SCHEMBL6644584

SCHEMBL6644584

CN1CCCC1c1nccc(C(N)=O)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.49
PARP2 Q9UGN5 1/20 0.42
KDM4E B2RXH2 1/20 0.41
BLM P54132 1/20 0.41
ALOX15 P16050 1/20 0.41
ALDH1A1 P00352 2/20 0.40
CHRNA7 P36544 2/20 0.40
CHRNB2 P17787 2/20 0.40
CHRNB4 P30926 2/20 0.40
CHRNA3 P32297 2/20 0.40
CHRNA4 P43681 2/20 0.40
CHRNA2 Q15822 2/20 0.40
LMNA P02545 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HTR3E A5X5Y0 1/20 0.40
PSIP1 O75475 1/20 0.40
TRPA1 O75762 1/20 0.40
HTR3B O95264 1/20 0.40
CHRNA1 P02708 1/20 0.40
CHRNG P07510 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6644661 0.83 PARP1 (0.37) PARP1PARP2
SCHEMBL10002467 0.75 ALDH1A1 (0.50) ALDH1A1CHRNA7CHRNB2CHRNB4CHRNA3
SCHEMBL1831858 0.74 ALOX5AP (0.43) KDM4ETDP1
SCHEMBL1833909 0.74 GSK3B (0.38) KDM4E
SCHEMBL13330409 0.73 CHRNB2 (0.53) ALDH1A1CHRNA7CHRNB2CHRNB4CHRNA3
SCHEMBL22720412 0.73 PARP1 (0.42) PARP1PARP2CHRNB4CHRNA3
SCHEMBL6185263 0.72 PARP1 (0.43) PARP1PARP2KDM4EBLMALOX15
SCHEMBL27797718 0.69 HRH3 (0.46) KDM4EALDH1A1MAPT
SCHEMBL6645725 0.69 PARP1 (0.45) PARP1PARP2CHRNA7CHRNB2CHRNA4
Acetic Acid SCHEMBL27199919 0.69 KDM4E (0.43) KDM4EBLMALOX15ALDH1A1CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441734-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2004-08-04 EP disclosed
WO-2003035076-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2003-05-01 WO disclosed