SCHEMBL6645319

SCHEMBL6645319

CS(=O)(=O)NCCCOc1ccc(N)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
KMT2A Q03164 3/20 0.56
HTT P42858 2/20 0.56
MEN1 O00255 2/20 0.56
PKM P14618 2/20 0.49
LMNA P02545 1/20 0.49
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
CYP4F2 P78329 1/20 0.46
CYP4A11 Q02928 1/20 0.46
TDP1 Q9NUW8 2/20 0.46
MAPT P10636 2/20 0.45
KDM4E B2RXH2 1/20 0.45
TSHR P16473 2/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14410510 0.85 DRD2 (0.61) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL4975281 0.84 ALDH1A1 (0.55) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL6645317 0.81 PARP10 (0.54) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL13301478 0.81 ALDH1A1 (0.62) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL13177810 0.81 ALDH1A1 (0.55) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL15904079 0.80 ALDH1A1 (0.54) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL13178011 0.80 ALDH1A1 (0.54) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL10191940 0.79 ALDH1A1 (0.65) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL10336962 0.79 ALDH1A1 (0.69) ALDH1A1KMT2AHTTMEN1PKM
SCHEMBL2227724 0.79 TDP1 (0.52) ALDH1A1KMT2ANPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453831-A1 1H-PYRROLO(3,2-B)PYRIDINE-3-CARBOXYLIC ACID AMIDES Neurogen Corporation (US) 2004-09-08 EP claimed
US-6673811-B1 TREATMENT OF ANXIETY, DEPRESSION, SLEEP DISORDER, ATTENTION DEFICIT DISORDER, ALZHEIMER'S DEMENTIA, OR SHORT-TERM MEMORY LOSS NEUROGEN CORPORATION 2004-01-06 US claimed
WO-2003044018-A1 1H-PYRROLO[3,2-B]PYRIDINE-3-CARBOXYLIC ACID AMIDES NEUROGEN CORPORATION (US) 2003-05-30 WO claimed
US-6673811-B1 TREATMENT OF ANXIETY, DEPRESSION, SLEEP DISORDER, ATTENTION DEFICIT DISORDER, ALZHEIMER'S DEMENTIA, OR SHORT-TERM MEMORY LOSS NEUROGEN CORPORATION 2004-01-06 US disclosed