SCHEMBL6645786

SCHEMBL6645786

CCC(CC)NC(=O)c1cc(C(=O)O)cc(-c2ncco2)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GLRA3 O75311 1/20 0.44
GLRB P48167 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.39
HTT P42858 1/20 0.39
TAS1R3 Q7RTX0 5/20 0.38
TAS1R1 Q7RTX1 5/20 0.38
BACE1 P56817 1/20 0.37
HDAC4 P56524 1/20 0.37
LTA4H P09960 5/20 0.36
HCAR3 P49019 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
CREBBP Q92793 1/20 0.35
TRPM4 Q8TD43 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6646087 0.90 GLRA3 (0.44) GLRA3GLRBSMN1; SMN2BACE1LTA4H
SCHEMBL19928407 0.79 GLRA3 (0.46) GLRA3GLRBHDAC4LTA4HHCAR3
SCHEMBL6648461 0.79 NAAA (0.46) GLRA3GLRBSMN1; SMN2HTTHCAR3
SCHEMBL20256885 0.77 GLRA3 (0.49) GLRA3GLRBHDAC4LTA4HCREBBP
SCHEMBL475508 0.77 GLRA3 (0.70) GLRA3GLRBHDAC4LTA4HTRPM4
SCHEMBL2207635 0.74 BACE1 (0.44) GLRA3GLRBSMN1; SMN2BACE1LTA4H
SCHEMBL15131324 0.74 GLRA3 (0.46) GLRA3GLRBHDAC4LTA4HTRPM4
SCHEMBL2908806 0.73 HTT (0.63) SMN1; SMN2HTTTAS1R3TAS1R1
Hydrochloric Acid SCHEMBL6172352 0.73 BACE1 (0.44) GLRA3GLRBSMN1; SMN2BACE1LTA4H
SCHEMBL3348971 0.73 GLRA3 (0.41) GLRA3GLRBBACE1LTA4HHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453789-A2 N,N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2004-09-08 EP disclosed
WO-2003040096-A2 N, N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2003-05-15 WO disclosed