SCHEMBL6652677

SCHEMBL6652677

Nc1ccc(Nc2ccc(C(=O)c3ccccc3)cc2)c(Cl)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.69
GAA P10253 3/20 0.69
TDP1 Q9NUW8 2/20 0.69
ALOX15 P16050 1/20 0.69
HTT P42858 1/20 0.69
MAPK13 O15264 5/20 0.61
MAPK12 P53778 5/20 0.61
MAPK11 Q15759 5/20 0.61
MAPK14 Q16539 5/20 0.61
MAPT P10636 3/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
HSD17B10 Q99714 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
KDM4E B2RXH2 2/20 0.50
DHODH Q02127 2/20 0.50
PBRM1 Q86U86 1/20 0.50
THRB P10828 1/20 0.50
HPGD P15428 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11798862 0.87 MAPK13 (0.72) ALDH1A1GAATDP1ALOX15HTT
SCHEMBL6656529 0.84 MAPK13 (0.60) ALDH1A1GAAMAPK13MAPK12MAPK11
SCHEMBL6656304 0.84 MAPT (0.61) ALDH1A1GAATDP1ALOX15HTT
SCHEMBL6653594 0.82 MAPK13 (0.70) ALDH1A1GAAALOX15HTTMAPK13
SCHEMBL15968528 0.82 GAA (1.00) ALDH1A1GAATDP1ALOX15HTT
SCHEMBL2789324 0.81 MAPK13 (0.78) ALDH1A1TDP1HTTMAPK13MAPK12
SCHEMBL2791237 0.81 MAPK13 (0.78) ALDH1A1TDP1HTTMAPK13MAPK12
SCHEMBL6655626 0.81 MAPK13 (0.56) ALDH1A1GAATDP1ALOX15HTT
SCHEMBL6657520 0.80 CTSV (0.56) ALDH1A1MAPK13MAPK12MAPK11MAPK14
SCHEMBL27483181 0.78 MAPK13 (0.64) ALDH1A1GAAALOX15MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1188388-C Aminobenzophenones as inhibitors of interleukin and TNF LEO PHARM PROD LTD (DK) 2005-02-09 CN disclosed
EP-0966424-B1 AMINOBENZOPHENONES AS INHIBITORS OF INTERLEUKIN AND TNF LEO PHARMA AS (DK) 2004-06-23 EP disclosed
US-6313174-B1 FOR THERAPY AND PROPHYLAXIS OF ASTHMA, ALLERGY, RHEUMATOID ARTHRITIS, SPONDYLOARTHRITIS, GOUT, ATHEROSCLEROSIS, CHRONIC INFLAMMATORY BOWEL DISEASE, PROLIFERATIVE AND INFLAMMATORY SKIN DISORDERS Leo Pharmaceutical Products Ltd.A/S/ (Løvens kemiske Fabrik Produktionsaktieselskab) (DK) 2001-11-06 US disclosed