SCHEMBL6652994

SCHEMBL6652994

CC(C)(C)C(N)C(=O)c1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP8 Q6V1X1 2/20 0.45
DPP9 Q86TI2 2/20 0.45
DPP4 P27487 1/20 0.45
DPP7 Q9UHL4 1/20 0.45
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
BCL2L1 Q07817 1/20 0.39
BAD Q92934 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39
KCNN4 O15554 1/20 0.38
PTPN1 P18031 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HTR7 P34969 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6652998 1.00 DPP8 (0.45) DPP8DPP9DPP4DPP7CES2
SCHEMBL6654144 0.82 PDPK1 (0.46) CES2CA1CA2SLC6A2SLC6A3
SCHEMBL6654142 0.82 PDPK1 (0.46) CES2CA1CA2SLC6A2SLC6A3
SCHEMBL16234935 0.81 TRPA1 (0.50) CES2CES1CA1CA2NPC1
Hydrochloric Acid SCHEMBL6462076 0.81 PDPK1 (0.44) CES2CA1CA2SLC6A2SLC6A3
SCHEMBL8251886 0.80 TDP1 (0.47) CES2CES1NPC1RAB9AMAPT
Hydrochloric Acid SCHEMBL16235165 0.79 TRPA1 (0.49) CES2CES1CA1CA2NPC1
SCHEMBL23571752 0.78 CES2 (0.46) CES2CES1CA1CA2SLC6A2
SCHEMBL10444348 0.78 CES2 (0.46) CES2CES1CA1CA2SLC6A2
SCHEMBL6653842 0.78 CA1 (0.53) CES2CES1CA1CA2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000061134-A9 ANTIMICROBIAL AGENTS BRITISH BIOTECH PHARM (GB) 2004-04-22 WO disclosed
US-6716878-B1 BACTERICIDE, ANTIPROTOZOAL; VANCOMYCIN RESISTANT ENTEROCOCCI AND BETA-LACTAM ANTIBIOTIC-RESISTANT BACTERIA, METHICILLIN-RESISTANT STAPHYLOCOCCUS AUREUS; HYDROXAMIC ACID AND N-FORMYL SUBTITUTED ALKYLAMIDES VERNALIS (OXFORD) LIMITED (GB) 2004-04-06 US disclosed
EP-1169031-A1 ANTIMICROBIAL AGENTS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 2002-01-09 EP disclosed
WO-2000061134-A1 ANTIMICROBIAL AGENTS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 2000-10-19 WO disclosed