SCHEMBL665777

SCHEMBL665777

[CH2]C(O)CN1CCOCC1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.67
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 3/20 0.47
ANPEP P15144 1/20 0.47
KDM4E B2RXH2 4/20 0.46
ATM Q13315 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
HSD17B10 Q99714 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP2D6 P10635 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL663967 1.00 USP2 (0.67) USP2MEN1KMT2AALDH1A1ANPEP
SCHEMBL665275 1.00 USP2 (0.67) USP2MEN1KMT2AALDH1A1ANPEP
SCHEMBL709506 0.80 USP2 (1.00) USP2MEN1KMT2AALDH1A1ANPEP
SCHEMBL13024067 0.80 USP2 (0.73) USP2MEN1KMT2AALDH1A1ANPEP
SCHEMBL22278256 0.80 USP2 (0.73) USP2MEN1KMT2AALDH1A1ANPEP
SCHEMBL4373095 0.77
SCHEMBL1829243 0.77
SCHEMBL4388841 0.77
SCHEMBL1504812 0.77
SCHEMBL24688084 0.76 USP2 (0.67) USP2MEN1KMT2AALDH1A1ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 169 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117062815-A VMAT2 inhibitors and methods of use 纽罗克里生物科学有限公司 2023-11-14 CN claimed
EP-4168409-A1 VMAT2 INHIBITORS AND METHODS OF USE Neurocrine Biosciences, Inc. (US) 2023-04-26 EP claimed
WO-2011033094-A1 SCHEDULE OF ADMINISTRATION OF BENZAZOLE DERIVATIVES IN THE TREATMENT OF LEUKEMIAS 4SC AG (DE) 2011-03-24 WO claimed
WO-2010110686-A1 PYRIMIDINYL AND 1,3,5 TRIAZINYL BENZIMIDAZOLES AND THEIR USE IN CANCER THERAPY PATHWAY THERAPEUTICS LIMITED (NZ) 2010-09-30 WO claimed
EP-1007530-B1 6-O-SUBSTITUTED ERYTHROMYCIN COMPOUNDS AND METHOD FOR MAKING SAME ABBOTT LAB (US) 2005-11-16 EP claimed
CN-1642949-A Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterial, related compositions and methods ORTHO MCNEIL PHARM INC (US) 2005-07-20 CN claimed
EP-1470123-A1 BICYCLIC HETEROCYCLIC SUBSTITUTED PHENYL OXAZOLIDINONE ANTIBACTERIALS, RELATED COMPOSITIONS AND METHODS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-10-27 EP claimed
US-20040067994-A1 BICYCLIC HETEROCYCLIC SUBSTITUTED PHENYL OXAZOLIDINONE ANTIBACTERIALS, AND RELATED COMPOSITIONS AND METHODS PAGET STEVEN D (US) 2004-04-08 US claimed
CN-1142912-C Amide derivs. useful as inhibitors of production of cytokines 2004-03-24 CN claimed
US-6608081-B2 Treating pneumonia ORTHO-MCNEIL PHARMACEUTICAL, INC. 2003-08-19 US claimed
CN-1224427-A 6-O-substituted erythromycin compounds and preparation method thereof ABBOTT LAB (US) 1999-07-28 CN claimed
EP-0918783-A1 6-O-SUBSTITUTED ERYTHROMYCINS AND METHOD FOR MAKING THEM ABBOTT LABORATORIES (US) 1999-06-02 EP claimed
EP-0679945-B1 Processing of a silver halide photgraphic with a peroxide bleach composition EASTMAN KODAK CO (US) 1998-08-19 EP claimed
WO-1997042206-A1 6-O-SUBSTITUTED ERYTHROMYCIN COMPOUNDS AND METHOD FOR MAKING SAME ABBOTT LABORATORIES (US) 1997-11-13 WO claimed
WO-1997042204-A1 6-O-SUBSTITUTED ERYTHROMYCINS AND METHOD FOR MAKING THEM ABBOTT LABORATORIES (US) 1997-11-13 WO claimed
EP-0679945-A2 Hydrogen peroxide bleach composition for use with silver halide photographic elements EASTMAN KODAK COMPANY (US) 1995-11-02 EP claimed
WO-1993024490-A1 USE OF INDOLOCARBAZOLS IN AIDS TREATMENT Gödecke Aktiengesellschaft (DE) 1993-12-09 WO claimed
EP-0370236-B1 INDOLOCARBAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS GÖDECKE AKTIENGESELLSCHAFT (DE) 1991-12-27 EP claimed
EP-0370236-A1 Indolocarbazole derivatives, processes for their preparation and their use as medicaments GÖDECKE AKTIENGESELLSCHAFT (DE) 1990-05-30 EP claimed
US-4801601-A ANTILEUKEMIA AGENT HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1989-01-31 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040067994-A1 BICYCLIC HETEROCYCLIC SUBSTITUTED PHENYL OXAZOLIDINONE ANTIBACTERIALS, AND RELATED COMPOSITIONS AND METHODS OXA1L, NDUFS3, CYCS USP2 4346/4885MEN1 4298/4885KMT2A 3290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.