SCHEMBL6658084

SCHEMBL6658084

CCN1CCCCC1C(=O)N1CCN(Cc2ccc(OC)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
POLB P06746 1/20 0.52
PKM P14618 1/20 0.52
ALDH1A1 P00352 1/20 0.49
FAAH O00519 1/20 0.49
HRH3 Q9Y5N1 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
SIGMAR1 Q99720 1/20 0.47
LSS P48449 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PTGIR P43119 1/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6658081 1.00 KDM4E (0.54) KDM4EPOLBPKMALDH1A1FAAH
Hydrochloric Acid SCHEMBL6663247 0.86 NPBWR1 (0.55) KDM4EPOLBALDH1A1HRH3L3MBTL1
SCHEMBL6659429 0.86 L3MBTL1 (0.50) L3MBTL1
Hydrochloric Acid SCHEMBL6663643 0.86 NPBWR1 (0.55) KDM4EPOLBALDH1A1HRH3L3MBTL1
SCHEMBL6908168 0.86 L3MBTL1 (0.50) L3MBTL1
SCHEMBL6663904 0.86 KMT2A (0.57) KDM4EPOLBALDH1A1HRH3L3MBTL1
SCHEMBL6905958 0.86 KMT2A (0.57) KDM4EPOLBALDH1A1HRH3L3MBTL1
SCHEMBL27506526 0.84 KDM4E (0.51) KDM4EPOLBALDH1A1L3MBTL1SMN1; SMN2
Hydrochloric Acid SCHEMBL6659280 0.83 KDM4E (0.50) KDM4EPOLBALDH1A1L3MBTL1SMN1; SMN2
Hydrochloric Acid SCHEMBL6659274 0.83 KDM4E (0.50) KDM4EPOLBALDH1A1L3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441728-A2 MODULATORS OF THE CHOLESTEROL BIOSYNTHETIC PATHWAY Vertex Pharmaceuticals Incorporated (US) 2004-08-04 EP disclosed
WO-2003037338-A2 MODULATORS OF THE CHOLESTEROL BIOSYNTHETIC PATHWAY VERTEX PHARMACEUTICALS INCORPORATED (US) 2003-05-08 WO disclosed
EP-1257544-A2 PIPERAZINE AND PIPERIDINE DERIVATIVES FOR TREATMENT OR PREVENTION OF NEURONAL DAMAGE Vertex Pharmaceuticals Incorporated (US) 2002-11-20 EP disclosed
WO-2001058891-A2 PIPERAZINE AND PIPERIDINE DERIVATIVES FOR TREATMENT OR PREVENTION OF NEURONAL DAMAGE VERTEX PHARMACEUTICALS INCORPORATED (US) 2001-08-16 WO disclosed