SCHEMBL6659233

SCHEMBL6659233

Fc1ccc(Oc2ncnc3[nH]cnc23)cc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 9/20 0.60
FLT3 P36888 1/20 0.44
TTBK1 Q5TCY1 1/20 0.44
TTBK2 Q6IQ55 1/20 0.44
MRGPRX1 Q96LB2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CDK1 P06493 1/20 0.37
CSF1R P07333 1/20 0.36
DRD1 P21728 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2623130 0.84 TRPA1 (0.58) TRPA1FLT3TTBK1TTBK2MRGPRX1
SCHEMBL1791375 0.82 MERTK (0.55) FLT3DRD1
SCHEMBL23069173 0.81 TRPA1 (0.41) TRPA1DRD1
SCHEMBL822148 0.81 ALDH1A1 (0.47) TRPA1FLT3TTBK1ALDH1A1KDM4E
SCHEMBL1791378 0.78 TRPA1 (0.40) TRPA1FLT3CSF1R
SCHEMBL5358444 0.78 TRPA1 (0.35) TRPA1
SCHEMBL7830504 0.75 JAK2 (0.42) TRPA1ALDH1A1KDM4EDRD1SMN1; SMN2
SCHEMBL2940695 0.72 PDPK1 (0.36) TRPA1
SCHEMBL14104450 0.72 MAPT (0.44) TRPA1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL23977400 0.71 HAO1 (0.47) TRPA1FLT3DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444982-A1 The use of purine derivatives as selective kinase inhibitors MERCKLE GMBH (DE) 2004-08-11 EP disclosed