SCHEMBL6660161

SCHEMBL6660161

Oc1ccc2nc(-c3ccccc3)cc(-c3ccccc3F)c2c1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 18/20 0.65
ESR2 Q92731 18/20 0.65
ESRRB O95718 6/20 0.50
ESRRA P11474 6/20 0.50
ELANE P08246 1/20 0.49
MEN1 O00255 1/20 0.45
NTSR1 P30989 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6663329 0.88 ESR1 (0.69) ESR1ESR2ESRRBESRRAELANE
SCHEMBL28252108 0.83 ACHE (0.54)
SCHEMBL6662078 0.82 ESR1 (0.73) ESR1ESR2ESRRBESRRAELANE
SCHEMBL8956150 0.82 MAPK1 (0.63) ESR1ESR2ELANE
SCHEMBL3927237 0.79 ESR1 (1.00) ESR1ESR2ESRRBESRRAELANE
SCHEMBL3929568 0.77 ESR1 (0.76) ESR1ESR2ESRRBESRRA
SCHEMBL13458667 0.76 MAP4K1 (0.46) MEN1KMT2A
SCHEMBL6665622 0.76 ESR1 (0.48) ESR1ESR2ESRRBESRRAMEN1
SCHEMBL6534483 0.75 ESR1 (0.84) ESR1ESR2ESRRBESRRAELANE
SCHEMBL6666467 0.74 TOP1 (0.44) ELANEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861864-B1 Method of preparation of polyquinolines HITACHI CHEMICAL CO LTD (JP) 2004-08-25 EP disclosed
EP-0861864-A2 Method of preparation of polyquinolines HITACHI CHEMICAL CO., LTD. (JP) 1998-09-02 EP disclosed
US-5786071-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-07-28 US disclosed
US-5723573-A ACETYLENIC END GROUPS HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-03-03 US disclosed
US-5648448-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1997-07-15 US disclosed