SCHEMBL6663329

SCHEMBL6663329

Oc1ccc2nc(-c3ccccc3F)cc(-c3ccccc3)c2c1

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.69
ESR2 Q92731 13/20 0.69
ELANE P08246 1/20 0.49
ESRRB O95718 2/20 0.43
ESRRA P11474 2/20 0.43
MEN1 O00255 2/20 0.43
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPK1 P28482 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
RECQL P46063 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALOX5 P09917 1/20 0.42
GAA P10253 1/20 0.42
GPR35 Q9HC97 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6660161 0.88 ESR1 (0.65) ESR1ESR2ELANEESRRBESRRA
SCHEMBL6667127 0.85 ESR1 (0.54) ESR1ESR2ELANEMEN1MAPT
SCHEMBL7610922 0.83 ACACA (0.53) ESR1ESR2MAPTMAPK1KDM4E
SCHEMBL6662078 0.82 ESR1 (0.73) ESR1ESR2ELANEESRRBESRRA
SCHEMBL8956454 0.82 MAPK1 (0.63) ESR1ESR2ELANEMEN1MAPT
SCHEMBL3927237 0.82 ESR1 (1.00) ESR1ESR2ELANEESRRBESRRA
SCHEMBL440455 0.76 MAP4K1 (0.49) ESR1ESR2MEN1KMT2AMAPK1
SCHEMBL6665622 0.76 ESR1 (0.48) ESR1ESR2ESRRBESRRAMEN1
SCHEMBL23674185 0.75 ESR2 (0.56) ESR1ESR2ELANEESRRBESRRA
SCHEMBL10612165 0.75 ADORA2A (0.47) ESR1ESR2MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861864-B1 Method of preparation of polyquinolines HITACHI CHEMICAL CO LTD (JP) 2004-08-25 EP disclosed
EP-0861864-A2 Method of preparation of polyquinolines HITACHI CHEMICAL CO., LTD. (JP) 1998-09-02 EP disclosed
US-5786071-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-07-28 US disclosed
US-5723573-A ACETYLENIC END GROUPS HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-03-03 US disclosed
US-5648448-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1997-07-15 US disclosed