SCHEMBL6661754

SCHEMBL6661754

Nc1ncnc2ncn(Cc3ccc(F)cc3)c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.56
PIK3CD O00329 2/20 0.44
PI4KA P42356 1/20 0.43
PI4K2B Q8TCG2 1/20 0.43
PI4K2A Q9BTU6 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
ADORA1 P30542 1/20 0.42
MET P08581 2/20 0.41
NSD2 O96028 1/20 0.41
NSD3 Q9BZ95 1/20 0.41
EGFR P00533 1/20 0.41
SRC P12931 1/20 0.41
KDR P35968 1/20 0.41
TEK Q02763 1/20 0.41
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
QPCT Q16769 2/20 0.39
QPCTL Q9NXS2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4343213 0.85 ADORA2A (0.60) ADORA2APIK3CDPI4KAPI4K2BPI4K2A
SCHEMBL6665170 0.84 MET (0.42) ADORA2AMETHTTSMN1; SMN2LMNA
SCHEMBL22533303 0.82 ADORA2A (0.52) ADORA2APIK3CDPI4KAPI4K2BPI4K2A
SCHEMBL29424717 0.82 ADORA2A (0.52) ADORA2APIK3CDPI4KAPI4K2BPI4K2A
Hydrochloric Acid SCHEMBL29424851 0.81 ADORA2A (0.51) ADORA2APIK3CDPI4KAPI4K2BPI4K2A
Hydrochloric Acid SCHEMBL22533583 0.81 ADORA2A (0.51) ADORA2APIK3CDPI4KAPI4K2BPI4K2A
SCHEMBL6662357 0.79 MET (0.47) ADORA2AMETHTTSMN1; SMN2CYP11B2
SCHEMBL6659204 0.77 ADORA2A (0.74) ADORA2API4KAPI4K2BPI4K2API4KB
SCHEMBL1665392 0.74 ADORA2A (0.71) ADORA2APIK3CDPI4KAPI4K2BPI4K2A
SCHEMBL21121650 0.73 ADORA2A (0.40) ADORA2API4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444982-A1 The use of purine derivatives as selective kinase inhibitors MERCKLE GMBH (DE) 2004-08-11 EP disclosed