SCHEMBL6662357

SCHEMBL6662357

COc1ncnc2ncn(Cc3ccc(F)cc3)c12

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MET P08581 3/20 0.47
KDM4E B2RXH2 4/20 0.42
HPGD P15428 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP11B2 P19099 2/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GAA P10253 2/20 0.38
TSHR P16473 1/20 0.38
CYP11B1 P15538 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPK14 Q16539 1/20 0.37
AURKA O14965 1/20 0.37
ACHE P22303 1/20 0.37
BACE1 P56817 1/20 0.37
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28663481 0.86 HPGD (0.52) HPGDALDH1A1CYP11B2SMN1; SMN2GAA
SCHEMBL29424821 0.83 HPGD (0.37) METHPGDGAAADORA2A
SCHEMBL22533657 0.83 HPGD (0.37) METHPGDGAAADORA2A
SCHEMBL6665170 0.80 MET (0.42) METKDM4EHPGDALDH1A1CYP11B2
SCHEMBL6661754 0.79 ADORA2A (0.56) METKDM4EALDH1A1CYP11B2HTT
SCHEMBL29434725 0.74 ALDH1A1 (0.52) METKDM4EHPGDALDH1A1CYP11B2
SCHEMBL20187539 0.74 ALDH1A1 (0.52) METKDM4EHPGDALDH1A1CYP11B2
SCHEMBL22221944 0.74 ADORA2A (0.62) ADORA2A
SCHEMBL21883518 0.72 MET (0.46) METKDM4EHPGDALDH1A1CYP11B2
SCHEMBL30021455 0.72 MET (0.46) METKDM4EHPGDALDH1A1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444982-A1 The use of purine derivatives as selective kinase inhibitors MERCKLE GMBH (DE) 2004-08-11 EP disclosed