SCHEMBL6662151

SCHEMBL6662151

Cc1c(C(F)(F)F)cc(C(=O)Nc2ccc3c(c2)CCN3C(=O)Cc2ccccn2)c(-c2ccccc2)c1C

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 13/20 0.48
HTR2C P28335 13/20 0.48
HTR2B P41595 12/20 0.48
EIF2AK3 Q9NZJ5 1/20 0.43
MTTP P55157 2/20 0.43
SMO Q99835 2/20 0.43
APOB P04114 1/20 0.43
CYP1A2 P05177 2/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6670014 0.90 EIF2AK3 (0.45) HTR2AHTR2CHTR2BEIF2AK3MTTP
SCHEMBL6667820 0.89 SMO (0.50) HTR2AHTR2CHTR2BEIF2AK3MTTP
SCHEMBL6669100 0.88 EIF2AK3 (0.45) HTR2AHTR2CHTR2BEIF2AK3MTTP
SCHEMBL6664165 0.87 EIF2AK3 (0.46) HTR2AHTR2CHTR2BEIF2AK3MTTP
SCHEMBL6667664 0.86 HTR2A (0.49) HTR2AHTR2CHTR2BEIF2AK3MTTP
SCHEMBL6799789 0.85 SMO (0.54) HTR2AHTR2CHTR2BEIF2AK3MTTP
SCHEMBL6665604 0.85 HTR2C (0.47) HTR2AHTR2CHTR2BEIF2AK3MTTP
SCHEMBL6666452 0.85 HTR2A (0.44) HTR2AHTR2CHTR2BEIF2AK3SMO
SCHEMBL6665112 0.85 HTR2C (0.46) HTR2AHTR2CHTR2BEIF2AK3SMO
SCHEMBL6665020 0.84 HTR2A (0.44) HTR2AHTR2CHTR2BEIF2AK3SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383760-A1 BIARYLCARBOXAMIDE COMPOUNDS AS APOLIPOPROTEIN B INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-01-28 EP disclosed
WO-2002090347-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-14 WO disclosed