SCHEMBL6662228

SCHEMBL6662228

CCN1C(=O)c2cc(Cl)ccc2C(C(=O)NC2CCCC2)C1c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 2/20 0.42
TACR1 P25103 2/20 0.42
ALDH1A1 P00352 2/20 0.40
GAA P10253 2/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
FFAR1 O14842 1/20 0.37
CETP P11597 3/20 0.37
TP53 P04637 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
MDM2 Q00987 1/20 0.37
RHOC P08134 1/20 0.36
RHOA P61586 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
ACKR3 P25106 1/20 0.36
EPHX2 P34913 1/20 0.36
CRHR1 P34998 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6417300 0.88 TACR2 (0.43) TACR2TACR1ALDH1A1CETPCNR1
SCHEMBL6410700 0.81 GAA (0.54) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL6412758 0.78 ALDH1A1 (0.56) ALDH1A1GAA
SCHEMBL6412106 0.76 GAA (0.46) ALDH1A1GAATP53
SCHEMBL6414932 0.76 MAPT (0.47) ALDH1A1GAANPC1FFAR1
SCHEMBL6417286 0.75 L3MBTL1 (0.49) ALDH1A1GAACNR2
SCHEMBL6412336 0.75 TSHR (0.63) ALDH1A1GAASMN1; SMN2TP53
SCHEMBL6417824 0.74 ALDH1A1 (0.50) ALDH1A1GAAFFAR1
SCHEMBL6413218 0.74 HSD17B10 (0.47) ALDH1A1GAANPC1FFAR1
SCHEMBL6419707 0.74 TSHR (0.43) ALDH1A1GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004004727-A1 3,4-DIHYDROISOQUINOLIN-1-ONE DERIVATIVES AS INDUCERS OF APOPTOSIS AXYS PHARMACEUTICALS, INC. (US) 2004-01-15 WO claimed