SCHEMBL6663342

SCHEMBL6663342

Cn1cnc2c(Sc3ccc(F)cc3)ncnc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.45
ADORA2A P29274 1/20 0.45
YTHDC1 Q96MU7 1/20 0.43
CDK1 P06493 1/20 0.38
SLC29A1 Q99808 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
PKM P14618 1/20 0.37
NFKB1 P19838 1/20 0.37
THPO P40225 1/20 0.37
PMP22 Q01453 1/20 0.37
TSHR P16473 1/20 0.37
NSD2 O96028 1/20 0.36
NSD3 Q9BZ95 1/20 0.36
MAPK14 Q16539 1/20 0.35
MAPT P10636 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6661513 0.85 SLC29A1 (0.49) ADORA1ADORA2AYTHDC1CDK1SLC29A1
SCHEMBL6664688 0.79 SLC29A1 (0.57) SLC29A1CYP1A2PKMTSHRHTT
SCHEMBL6660729 0.78 SLC29A1 (0.59) ADORA2ASLC29A1
SCHEMBL6659707 0.75 ADORA2A (0.55) ADORA2ASLC29A1CYP1A2HTT
SCHEMBL31060261 0.75 ADORA2A (0.55) ADORA2ASLC29A1CYP1A2HTT
SCHEMBL6426384 0.74 CYP1A2 (0.59) ADORA1ADORA2AYTHDC1CDK1CYP1A2
SCHEMBL6663756 0.74 ADORA1 (0.49) ADORA1ADORA2AYTHDC1CDK1CYP1A2
SCHEMBL6666118 0.72 SLC29A1 (0.56) ADORA2ASLC29A1CYP1A2HTT
SCHEMBL31061437 0.72 SLC29A1 (0.56) ADORA2ASLC29A1CYP1A2HTT
SCHEMBL6660434 0.72 ADORA3 (0.55) ADORA1ADORA2AMAPK14MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444982-A1 The use of purine derivatives as selective kinase inhibitors MERCKLE GMBH (DE) 2004-08-11 EP disclosed