SCHEMBL6663728

SCHEMBL6663728

Cn1c(-c2ccc([S+](C)[O-])cc2)nc2c(Sc3ccccc3)ncnc21

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 16/20 0.48
ADORA1 P30542 16/20 0.48
ADORA2A P29274 15/20 0.48
ADORA2B P29275 9/20 0.48
PI4KA P42356 1/20 0.48
PI4K2B Q8TCG2 1/20 0.48
PI4K2A Q9BTU6 1/20 0.48
PI4KB Q9UBF8 1/20 0.48
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
CDK2 P24941 1/20 0.33
PLK1 P53350 1/20 0.33
BTK Q06187 1/20 0.33
ITK Q08881 1/20 0.33
IKBKE Q14164 1/20 0.33
SLC29A1 Q99808 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665550 0.89 ADORA3 (0.45) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6660016 0.87 ADORA3 (0.62) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6660810 0.84 ADORA3 (0.52) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6667230 0.82 ADORA3 (0.48) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6660434 0.79 ADORA3 (0.55) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6662360 0.77 ADORA3 (0.46) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6661208 0.74 MAPK13 (0.50) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL19103227 0.67 HPGD (0.40)
SCHEMBL4064829 0.66 ADORA2A (1.00) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL783764 0.66 ADORA3 (0.68) ADORA3ADORA1ADORA2AADORA2BPI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444982-A1 The use of purine derivatives as selective kinase inhibitors MERCKLE GMBH (DE) 2004-08-11 EP disclosed