SCHEMBL6661208

SCHEMBL6661208

CSc1ccc(-c2nc3c(Sc4ccc(F)cc4)ncnc3n2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 7/20 0.50
MAPK12 P53778 7/20 0.50
MAPK11 Q15759 7/20 0.50
MAPK14 Q16539 7/20 0.50
GCGR P47871 4/20 0.50
ADORA3 P0DMS8 10/20 0.49
ADORA1 P30542 10/20 0.49
ADORA2A P29274 9/20 0.49
ADORA2B P29275 4/20 0.42
PI4KA P42356 1/20 0.42
PI4K2B Q8TCG2 1/20 0.42
PI4K2A Q9BTU6 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
LCK P06239 1/20 0.36
RET P07949 1/20 0.36
ALOX5 P09917 1/20 0.36
PRKACA P17612 1/20 0.36
RPS6KB1 P23443 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6660810 0.89 ADORA3 (0.52) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL6660434 0.89 ADORA3 (0.55) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL6660416 0.85 PTGS2 (0.46) ADORA3ADORA1ADORA2A
SCHEMBL6665550 0.85 ADORA3 (0.45) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL6660016 0.80 ADORA3 (0.62) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6659013 0.77 ADORA3 (0.48) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL4066247 0.74 ADORA3 (0.57) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6667230 0.74 ADORA3 (0.48) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6663728 0.74 ADORA3 (0.48) ADORA3ADORA1ADORA2AADORA2BPI4KA
SCHEMBL6663342 0.71 ADORA1 (0.45) MAPK14ADORA1ADORA2ACYP1A2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444982-A1 The use of purine derivatives as selective kinase inhibitors MERCKLE GMBH (DE) 2004-08-11 EP disclosed