SCHEMBL6663735

SCHEMBL6663735

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)OCCNc1cccc2c1C(=O)c1ccccc1C2=O

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.48
CTSK P43235 3/20 0.48
CTSB P07858 2/20 0.48
CTSL P07711 2/20 0.48
EPHX2 P34913 1/20 0.47
AKT1 P31749 1/20 0.47
ACE P12821 1/20 0.46
KLK5 Q9Y337 1/20 0.46
CCKAR P32238 4/20 0.45
CCKBR P32239 4/20 0.45
APP P05067 1/20 0.44
SCN9A Q15858 1/20 0.44
ATM Q13315 1/20 0.42
PARP1 P09874 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665187 0.95 CTSS (0.45) CTSSCTSKCTSBCTSLEPHX2
SCHEMBL6660460 0.95 CTSS (0.45) CTSSCTSKCTSBCTSLEPHX2
SCHEMBL6662292 0.94 CTSS (0.46) CTSSCTSKCTSBCTSLEPHX2
SCHEMBL6661594 0.94 CTSS (0.46) CTSSCTSKCTSBCTSLEPHX2
SCHEMBL6663550 0.87 ITGB3 (0.46) CTSSCTSKEPHX2AKT1KLK5
SCHEMBL6662026 0.85 MALT1 (0.45) EPHX2
SCHEMBL6658627 0.85 MALT1 (0.45) EPHX2
SCHEMBL6659896 0.84 MALT1 (0.44) KLK5APP
SCHEMBL6664650 0.84 MALT1 (0.44) KLK5APP
SCHEMBL6663606 0.83 MAPT (0.45) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087935-B1 ANTHRACENE DERIVATIVES AS ANTI-CANCER AGENTS BTG INT LTD (GB) 2004-08-18 EP disclosed