SCHEMBL6663786

SCHEMBL6663786

COc1ccc(OC(NC2CCC(c3ncnc4scc(-c5ccccc5)c34)CC2)C(C)O)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.45
ADRB3 P13945 9/20 0.45
ADRB1 P08588 8/20 0.45
MAPT P10636 4/20 0.44
LMNA P02545 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 2/20 0.43
TP53 P04637 1/20 0.43
FGFR1 P11362 2/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A1 P68400 1/20 0.40
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6662638 0.89 ADRB2 (0.43) ADRB2ADRB3ADRB1MAPTLMNA
SCHEMBL6663781 0.82 ADRB3 (0.63) ADRB2ADRB3ADRB1
SCHEMBL6662634 0.74 ADRB2 (0.60) ADRB2ADRB3ADRB1
SCHEMBL4441119 0.72 ADRB3 (0.70) ADRB2ADRB3ADRB1
SCHEMBL6667655 0.72 POLB (0.42) ADRB2ADRB3ADRB1MAPTLMNA
SCHEMBL6667635 0.71 ADRB2 (0.62) ADRB2ADRB3ADRB1
SCHEMBL6684421 0.69 ADRB3 (0.84) ADRB2ADRB3ADRB1
SCHEMBL6662632 0.66 ADRB3 (0.39) ADRB2ADRB3ADRB1MAPTLMNA
SCHEMBL31462338 0.66 FGFR1 (0.53) LMNAHPGDPOLBFGFR1KMT2A
SCHEMBL6667652 0.66 ADRB3 (0.50) ADRB2ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014850-A2 SUBSTITUTED AMINOPYRIMIDINES AS NEUROKININ ANTAGONISTS PREDIX PHARMACEUTICALS HOLDINGS, INC. (US) 2004-02-19 WO claimed
WO-2004014850-A2 SUBSTITUTED AMINOPYRIMIDINES AS NEUROKININ ANTAGONISTS PREDIX PHARMACEUTICALS HOLDINGS, INC. (US) 2004-02-19 WO disclosed