SCHEMBL6664525

SCHEMBL6664525

O=C1N[C@H](c2cc(C(F)(F)F)cc(C(F)(F)F)c2)C(C(=O)O)c2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.38
HSD17B10 Q99714 1/20 0.37
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
TNKS2 Q9H2K2 1/20 0.35
P2RX1 P51575 1/20 0.35
FFAR1 O14842 1/20 0.35
GALR3 O60755 1/20 0.35
ALDH1A1 P00352 1/20 0.35
STING1 Q86WV6 1/20 0.35
CETP P11597 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6410861 1.00 TACR1 (0.38) TACR1HSD17B10EDNRBEDNRAMEN1
SCHEMBL6410860 1.00 TACR1 (0.38) TACR1HSD17B10EDNRBEDNRAMEN1
SCHEMBL6418985 0.84 TACR1 (0.44) TACR1MEN1KMT2AATMALDH1A1
SCHEMBL671559 0.82 HSD17B10 (0.45) HSD17B10EDNRBEDNRATNKS2FFAR1
SCHEMBL671560 0.82 HSD17B10 (0.45) HSD17B10EDNRBEDNRATNKS2FFAR1
SCHEMBL671561 0.82 HSD17B10 (0.45) HSD17B10EDNRBEDNRATNKS2FFAR1
SCHEMBL6411515 0.81 TSHR (0.40) TACR1
SCHEMBL6414378 0.81 CYP2C19 (0.41) TACR1HSD17B10
SCHEMBL6417317 0.79 MAPT (0.47) TACR1MEN1KMT2AALDH1A1
SCHEMBL6415621 0.78 P2RX7 (0.39) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004004727-A1 3,4-DIHYDROISOQUINOLIN-1-ONE DERIVATIVES AS INDUCERS OF APOPTOSIS AXYS PHARMACEUTICALS, INC. (US) 2004-01-15 WO disclosed