SCHEMBL6665358

SCHEMBL6665358

COc1cc(-c2ccccc2)ccc1S(=O)(=O)Nc1cc(C)on1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.65
MAPK1 P28482 1/20 0.65
ACLY P53396 4/20 0.50
HPGD P15428 2/20 0.50
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
BRD4 O60885 2/20 0.47
BRD2 P25440 2/20 0.47
BRD3 Q15059 2/20 0.47
ALPL P05186 1/20 0.47
ALDH1A1 P00352 1/20 0.47
PKM P14618 1/20 0.47
SCN9A Q15858 1/20 0.46
PPIA P62937 1/20 0.46
ALOX12 P18054 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6666797 0.86 TSHR (0.60) TSHRMAPK1ACLYHPGDALPL
SCHEMBL6669808 0.85 TSHR (0.71) TSHRMAPK1HPGDCYP2C9ALDH1A1
SCHEMBL23440286 0.79 TSHR (1.00) TSHRMAPK1CYP1A2CYP2C9ALDH1A1
SCHEMBL21609152 0.78 KAT6A (0.65) ACLYBRD4ALPL
SCHEMBL23440311 0.77 TSHR (0.80) TSHRMAPK1CYP1A2CYP2C9ALDH1A1
SCHEMBL1027519 0.73 TSHR (0.83) TSHRMAPK1CYP1A2CYP2C9ALDH1A1
SCHEMBL5183416 0.71 ALDH1A1 (0.61) TSHRMAPK1CYP2C9ALDH1A1PPIA
SCHEMBL23440280 0.71 TSHR (0.68) TSHRMAPK1ACLYHPGDCYP2C9
SCHEMBL6667306 0.71 MAPK1 (0.76) TSHRMAPK1CYP2C9ALDH1A1PPIA
SCHEMBL23440297 0.71 TSHR (0.75) TSHRMAPK1CYP1A2CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004021997-A2 INHIBITORS OF FUNGAL INVASION MICROBIA, INC. (US) 2004-03-18 WO disclosed