SCHEMBL6665647

SCHEMBL6665647

Cc1ccc2c(n1)NC(=O)C21CCCN(C(=O)O)C1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.38
PROKR1 Q8TCW9 1/20 0.32
PDE5A O76074 2/20 0.32
PIK3CD O00329 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MEN1 O00255 1/20 0.30
PKM P14618 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP3A4 P08684 1/20 0.30
HIF1A Q16665 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6637338 0.79 HTR1A (0.36) MAPK14PDE5APIK3CD
Hydrochloric Acid SCHEMBL6642177 0.78 HTR1A (0.36) MAPK14PDE5APIK3CD
SCHEMBL6638001 0.71
SCHEMBL6875654 0.70 HTR1A (0.43) MEN1KMT2A
SCHEMBL23778423 0.68 HRH3 (0.37) MAPK14
SCHEMBL31536104 0.65 HTR1A (0.54)
SCHEMBL28978269 0.65 OPRM1 (0.33)
SCHEMBL21904278 0.65 IP6K1 (0.42) MAPK14CYP3A4
SCHEMBL28978271 0.64 CRBN (0.34)
SCHEMBL18850849 0.64 MARK3 (0.44) MAPK14PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1426375-A2 Analgesic spiroindole derivatives AstraZeneca AB (SE) 2004-06-09 EP disclosed
EP-1202994-B1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2004-04-14 EP disclosed
EP-1202994-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-05-08 EP disclosed
WO-2001005790-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2001-01-25 WO disclosed