SCHEMBL6666099

SCHEMBL6666099

Cc1ccc2ncnc(Nc3ccccc3O)c2c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.68
MAPK1 P28482 2/20 0.66
KDM4E B2RXH2 1/20 0.66
RET P07949 6/20 0.64
RAF1 P04049 5/20 0.63
BRAF P15056 5/20 0.63
NCOA1 Q15788 2/20 0.59
NCOA3 Q9Y6Q9 2/20 0.59
GAA P10253 2/20 0.59
MAPT P10636 3/20 0.56
LMNA P02545 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
KIF5B P33176 4/20 0.54
MEN1 O00255 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5564490 0.89 HTT (0.61) HTTMAPK1KDM4ERETRAF1
SCHEMBL5569001 0.83 EGFR (0.60) HTTMAPK1KDM4ERETNCOA1
SCHEMBL14511293 0.83 NCOA1 (0.61) HTTMAPK1KDM4ERAF1BRAF
SCHEMBL6662890 0.82 SMN1; SMN2 (0.74) HTTMAPK1KDM4ENCOA1NCOA3
SCHEMBL29236749 0.82 ABCG2 (0.62) HTTMAPK1RETRAF1BRAF
SCHEMBL6662659 0.81 HTT (0.67) HTTMAPK1KDM4ERAF1BRAF
SCHEMBL5564779 0.81 HTT (0.64) HTTMAPK1KDM4ERETRAF1
SCHEMBL6664779 0.80 HTT (0.64) HTTMAPK1KDM4ENCOA1NCOA3
SCHEMBL5564611 0.80 KDR (0.71) HTTMAPK1KDM4ERAF1BRAF
SCHEMBL2101381 0.80 HTT (1.00) HTTMAPK1KDM4ERETRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004013091-A2 4-ANILIDO SUBSTITUTED QUINAZOLINES AND USE THEREOF AS INHIBITORS OF EPIDERMAL GROWTH FACTOR RECEPTOR KINASES YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2004-02-12 WO disclosed