SCHEMBL6666490

SCHEMBL6666490

NC(=O)Oc1cnc(Cl)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SCN9A Q15858 3/20 0.41
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
CYP1A2 P05177 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
MPO P05164 1/20 0.33
TPO P07202 1/20 0.33
EPX P11678 1/20 0.33
LPO P22079 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18770225 0.82 MEN1 (0.40) MEN1KMT2ASCN9ACDK8TDP1
SCHEMBL29177384 0.82 KMT2A (0.40) MEN1KMT2ACHRNB2CHRNA4CCNC
SCHEMBL361444 0.81 ALDH1A1 (0.47) MEN1KMT2ASCN9ACHRNB2CHRNA4
SCHEMBL28903825 0.80 MEN1 (0.38) MEN1KMT2ACHRNB2CHRNA4
SCHEMBL28707710 0.78 PIK3CD (0.47) MEN1KMT2ACDK8
SCHEMBL28724684 0.76 MEN1 (0.43) MEN1KMT2ACDK8CYP1A2MPO
SCHEMBL28324875 0.76 SCN9A (0.37) MEN1KMT2ASCN9A
SCHEMBL28550715 0.76 MAPK1 (0.38) MEN1KMT2A
SCHEMBL28595145 0.76 ALDH1A1 (0.39) MEN1KMT2A
SCHEMBL27711610 0.72 NAPRT (0.46) MEN1KMT2ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117957227-A Pyridodiazepine derivatives as GABA Aγ1 PAM 豪夫迈·罗氏有限公司 2024-04-30 CN disclosed
EP-1458684-A2 THERAPEUTIC HETEROCYCLES AstraZeneca AB (SE) 2004-09-22 EP disclosed
WO-2003051276-A2 THERAPEUTIC HETEROCYCLES ASTRAZENECA AB (SE) 2003-06-26 WO disclosed