SCHEMBL6667466

SCHEMBL6667466

O=C(Nc1[c]c(Oc2nccc3cnccc23)ccc1)Nc1ccccc1S(=O)(=O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 15/20 0.40
IMPDH2 P12268 2/20 0.37
KCNA5 P22460 1/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
BLM P54132 1/20 0.36
KMT2A Q03164 1/20 0.36
NAMPT P43490 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5259740 0.80 TRPV1 (0.41) TRPV1KCNA5MEN1KMT2ANAMPT
SCHEMBL6681376 0.76 TRPV1 (0.42) TRPV1KCNA5MAPK1NAMPT
SCHEMBL5259747 0.76 MEN1 (0.43) TRPV1KCNA5MEN1KMT2A
SCHEMBL5259734 0.76 MEN1 (0.43) TRPV1KCNA5MEN1KMT2A
SCHEMBL5262987 0.74 TRPV1 (0.44) TRPV1KCNA5
SCHEMBL5262991 0.74 TRPV1 (0.44) TRPV1KCNA5
SCHEMBL5262880 0.69 MEN1 (0.46) MEN1KMT2ANAMPT
SCHEMBL5261648 0.69 MEN1 (0.46) MEN1KMT2ANAMPT
SCHEMBL5259289 0.68 CA12 (0.42) TRPV1MEN1KMT2A
SCHEMBL5259291 0.68 CA12 (0.42) TRPV1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383750-A2 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS Almirall Prodesfarma, S.A. (ES) 2004-01-28 EP disclosed
WO-2002057242-A2 UREA DERIVATIVES AS INTEGRIN ALPHA 4 ANTAGONISTS ALMIRALL PRODESFARMA, S.A. (ES) 2002-07-25 WO disclosed