SCHEMBL6669756

SCHEMBL6669756

NC(=O)N1C=Cc2ccccc2S1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
SCN4A P35499 1/20 0.42
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
BCHE P06276 2/20 0.41
ACHE P22303 1/20 0.41
P2RX4 Q99571 4/20 0.34
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
GRIN1 Q05586 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2B Q13224 1/20 0.30
NOX1 Q9Y5S8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7182054 0.84 P2RX4 (0.33) MAPK1LMNATSHRSCN4ASCN5A
SCHEMBL28782453 0.71 NPC1 (0.42) MAPK1LMNATSHRSCN4ASCN5A
SCHEMBL3017720 0.71
SCHEMBL11708478 0.71
SCHEMBL27462081 0.70 CA12 (0.41) LMNAALDH1A1
SCHEMBL4753850 0.69 TSHR (0.50) MAPK1LMNATSHRSCN4ASCN5A
SCHEMBL28896768 0.67 MAOA (0.35)
SCHEMBL25197006 0.67
SCHEMBL31499308 0.66 MTNR1A (0.42) MAPK1BCHEGAANOX1
SCHEMBL9661765 0.64 SCN2A (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1688315-A Use of selective COX-2 inhibitors for the treatment of urinary incontinence RECORDATI S P A (CH) 2005-10-26 CN claimed
WO-2004019933-A1 METHOD OF PREVENTING OR TREATING ATHEROSCLEROSIS OR RESTENOSIS PHARMACIA & UPJOHN COMPANY (US) 2004-03-11 WO claimed
EP-3921623-A1 METHOD OF TESTING CRYSTALLINITY IN AMORPHOUS PHARMACEUTICAL COMPOSITIONS ColVisTec AG (DE) 2021-12-15 EP disclosed
CN-113424045-A Method for testing crystallinity in amorphous pharmaceutical compositions 科尔维斯科技股份公司 2021-09-21 CN disclosed
WO-2020160980-A1 METHOD OF TESTING CRYSTALLINITY IN AMORPHOUS PHARMACEUTICAL COMPOSITIONS COLVISTEC AG (DE) 2020-08-13 WO disclosed
CN-109369639-A A kind of purification process of piroxicam 重庆三圣实业股份有限公司 2019-02-22 CN disclosed
CN-102307857-A High penetration compositions and their use CHONGXI YU 2012-01-04 CN disclosed
CN-102264349-A Sphingolipid activator protein C and related protein and peptide fusogenic properties for transmembrane drug delivery systems 2011-11-30 CN disclosed
CN-1233323-C Orally disintegrating tablet of meloxicam and its preparation CHENGDU SHENGNUO SCIENCE AND T (CN) 2005-12-28 CN disclosed
CN-1658903-A Combinations of peroxisome proliferator-activated receptor (ppar) activator(s) and sterol absorption inhibitor(s) and treatments for vascular indications SCHERING CORP (US) 2005-08-24 CN disclosed
CN-1546033-A Orally disintegrating tablet of meloxicam and its preparation 成都圣诺科技发展有限公司 2004-11-17 CN disclosed
WO-2000071528-A1 4H-1,4-BENZOTHIAZINE-2-CARBOXAMIDES AND THEIR USE AS GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2000-11-30 WO disclosed
EP-0938477-A4 BENZOTHIAZO AND RELATED HETEROCYCLIC GROUP-CONTAINING CYSTEINE AND SERINE PROTEASE INHIBITORS CEPHALON INC (US) 1999-12-29 EP disclosed
EP-0938477-A1 BENZOTHIAZO AND RELATED HETEROCYCLIC GROUP-CONTAINING CYSTEINE AND SERINE PROTEASE INHIBITORS CEPHALON, INC. (US) 1999-09-01 EP disclosed
WO-1998021186-A1 BENZOTHIAZO AND RELATED HETEROCYCLIC GROUP-CONTAINING CYSTEINE AND SERINE PROTEASE INHIBITORS CEPHALON, INC. (US) 1998-05-22 WO disclosed
CN-1007893-B Process for preparation of ether matrix of anti-inflammatory oxacikam PFIZER (US) 1990-05-09 CN disclosed
CN-85102030-A The preparation method of the ethers parent medicine of antiphlogiston  Xi Kamu 1987-01-31 CN disclosed
CN-86103603-A The preparation method of the derivative of benzothiazine dioxide 1987-01-21 CN disclosed
CN-86103603-A The preparation method of the derivative of benzothiazine dioxide 1987-01-21 CN disclosed
EP-0034270-A1 Combinations of agents which give enhanced anti-inflammatory activity AMERICAN CYANAMID COMPANY (US) 1981-08-26 EP disclosed