SCHEMBL6670243

SCHEMBL6670243

COC(=O)CC(NC(=O)CN)c1ccc(-c2cccc(F)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.46
CTSA P10619 1/20 0.43
MME P08473 2/20 0.43
MMEL1 Q495T6 1/20 0.43
TAAR1 Q96RJ0 2/20 0.42
GPR34 Q9UPC5 1/20 0.41
TACR3 P29371 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
DCAF1 Q9Y4B6 1/20 0.40
PDE2A O00408 1/20 0.39
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
ACE P12821 1/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
POLB P06746 1/20 0.38
LGMN Q99538 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7172249 0.99 FFAR1 (0.45) FFAR1CTSAMMEMMEL1TAAR1
SCHEMBL6671291 0.89 TACR3 (0.41) CTSAGPR34TACR3DCAF1POLB
SCHEMBL6668894 0.88 HTT (0.47) FFAR1CTSATACR3MEN1KMT2A
Hydrochloric Acid SCHEMBL7171223 0.88 TACR3 (0.40) CTSATACR3DCAF1
Hydrochloric Acid SCHEMBL7170943 0.87 HTT (0.46) FFAR1CTSATACR3MEN1KMT2A
SCHEMBL6667674 0.87 MEN1 (0.51) CTSATACR3MEN1KMT2APOLB
SCHEMBL6667661 0.86 FFAR1 (0.46) FFAR1CTSAMMEMMEL1TAAR1
Hydrochloric Acid SCHEMBL7176606 0.86 MEN1 (0.50) CTSATACR3MEN1KMT2APOLB
Hydrochloric Acid SCHEMBL7177344 0.85 FFAR1 (0.45) FFAR1CTSAMMEMMEL1TAAR1
SCHEMBL18404162 0.84 ALDH1A1 (0.50) FFAR1CTSAMEN1KMT2ADCAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153014-B1 BETA-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2004-09-22 EP disclosed
EP-1153014-A2 BETA-ALANINE DERIVATIVES MERCK PATENT GmbH (DE) 2001-11-14 EP disclosed
WO-2000048996-A2 β-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2000-08-24 WO disclosed