SCHEMBL6671291

SCHEMBL6671291

COC(=O)CC(NC(=O)CN)c1cccc(-c2ccc(F)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.41
CTSA P10619 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
HTT P42858 1/20 0.39
ROCK2 O75116 4/20 0.39
ROCK1 Q13464 3/20 0.39
CHEK1 O14757 1/20 0.39
RPS6KA5 O75582 1/20 0.39
MAP4K4 O95819 1/20 0.39
CHEK2 O96017 1/20 0.39
PRKCG P05129 1/20 0.39
CDK1 P06493 1/20 0.39
PRKACA P17612 1/20 0.39
RPS6KB1 P23443 1/20 0.39
CDK2 P24941 1/20 0.39
MAPK1 P28482 1/20 0.39
AKT1 P31749 1/20 0.39
AKT2 P31751 1/20 0.39
GSK3A P49840 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7171223 0.99 TACR3 (0.40) TACR3CTSAALDH1A1MAPTHTT
SCHEMBL6670243 0.89 FFAR1 (0.46) TACR3CTSADCAF1POLBGPR34
SCHEMBL6668894 0.88 HTT (0.47) TACR3CTSAALDH1A1MAPTHTT
Hydrochloric Acid SCHEMBL7172249 0.88 FFAR1 (0.45) TACR3CTSADCAF1GPR34
Hydrochloric Acid SCHEMBL7170943 0.87 HTT (0.46) TACR3CTSAALDH1A1MAPTHTT
SCHEMBL18404162 0.84 ALDH1A1 (0.50) CTSAALDH1A1MAPTHTTDCAF1
SCHEMBL6670155 0.83 ALDH1A1 (0.41) CTSAALDH1A1MAPTHTTROCK2
Hydrochloric Acid SCHEMBL7171178 0.82 ALDH1A1 (0.40) CTSAALDH1A1MAPTHTTROCK2
SCHEMBL24036950 0.82 TACR3 (0.39) TACR3MAPTROCK2ROCK1CHEK1
SCHEMBL6667661 0.82 FFAR1 (0.46) TACR3CTSAMAPTDCAF1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153014-B1 BETA-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2004-09-22 EP disclosed
EP-1153014-A2 BETA-ALANINE DERIVATIVES MERCK PATENT GmbH (DE) 2001-11-14 EP disclosed
WO-2000048996-A2 β-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2000-08-24 WO disclosed