SCHEMBL6670720

SCHEMBL6670720

O=C(O)CCCCNc1ncccn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
HPGD P15428 1/20 0.51
ITGB3 P05106 2/20 0.47
ITGAV P06756 2/20 0.47
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
MAPK1 P28482 1/20 0.43
CDC25A P30304 1/20 0.43
CDC25B P30305 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TBXA2R P21731 1/20 0.42
PRMT1 Q99873 1/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
GFER P55789 1/20 0.42
HSD17B10 Q99714 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848939 0.94 ALDH1A1 (0.56) ALDH1A1HPGDITGB3ITGAVCDC25A
Trifluoroacetic Acid SCHEMBL6496568 0.91 ALDH1A1 (0.44) ALDH1A1HPGDITGB3ITGAVCYP1A2
SCHEMBL17234481 0.86 ALDH1A1 (0.60) ALDH1A1HPGDKMT2AKDM4EMEN1
SCHEMBL10767538 0.82 MAPK1 (0.49) ALDH1A1CYP1A2CYP2C9CYP2C19MAPK1
SCHEMBL3148784 0.80 KMT2A (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19MAPK1
SCHEMBL18794901 0.80 ALDH1A1 (0.52) ALDH1A1HPGDITGB3ITGAVCYP1A2
SCHEMBL2037116 0.80 ITGB3 (0.70) ITGB3ITGAV
SCHEMBL3135531 0.79 PRMT1 (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19MAPK1
SCHEMBL8501601 0.79 PRMT1 (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19MAPK1
SCHEMBL284282 0.79 PRMT1 (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153014-B1 BETA-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2004-09-22 EP disclosed
CN-1146541-C Beta-alanine derivatives Ĭ��ר���ɷ����޹�˾ 2004-04-21 CN disclosed
US-6576637-B1 Such as 3-(4-methyl-3-nitrophenyl)-3-(2-(4-(pyridin-2-yl-amino)butyryl amino)acetylamino)propionic acid; thrombosis, heart infarct, coronary heart diseases, arteriosclerosis, inflammations, MERCK PATENT GMBH (DE) 2003-06-10 US disclosed
CN-1340046-A Beta-alanine derivatives MERCK PATENT GMBH (DE) 2002-03-13 CN disclosed