SCHEMBL6670971

SCHEMBL6670971

COc1cccc(CC(=O)C(=O)O)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTBP2 P56545 1/20 0.68
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
CYP1A2 P05177 1/20 0.56
USP2 O75604 1/20 0.54
LMNA P02545 1/20 0.51
ALDH1A1 P00352 1/20 0.51
HTT P42858 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
MMP13 P45452 1/20 0.51
POLB P06746 1/20 0.51
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50
IDO1 P14902 1/20 0.50
AGXT P21549 1/20 0.50
RAB9A P51151 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
PTGS1 P23219 1/20 0.50
AKR1C3 P42330 1/20 0.50
AKR1C2 P52895 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9504420 0.90 CTBP2 (0.57) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL29824310 0.86 PTGS1 (0.67) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL229067 0.86 PTGS1 (0.67) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL7638956 0.85 CTBP2 (0.57) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL8218805 0.84 CTBP2 (0.65) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL8218798 0.84 CTBP2 (0.60) CTBP2MEN1KMT2ACYP1A2USP2
Hydrochloric Acid SCHEMBL8693464 0.84 CTBP2 (0.65) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL4071390 0.84 CTBP2 (0.64) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL7293162 0.83 CTBP2 (0.64) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL16902814 0.83 SMN1; SMN2 (0.53) CTBP2MEN1KMT2ALMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12428403-B2 N-(heterocyclyl and heterocyclylalkyl)-3-benzylpyridin-2-amine derivatives as SSTR4 agonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2025-09-30 US disclosed
CN-115485273-B N- (heterocyclyl and heterocyclylalkyl) -3-benzyl pyridin-2-amine derivatives as SSTR4 agonists 武田药品工业株式会社 2024-08-13 CN disclosed
US-20230192659-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-06-22 US disclosed
EP-4126849-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS Takeda Pharmaceutical Company Limited (JP) 2023-02-08 EP disclosed
CN-115485273-A N- (heterocyclyl and heterocyclylalkyl) -3-benzylpyridin-2-amine derivatives as SSTR4 agonists 武田药品工业株式会社 2022-12-16 CN disclosed
WO-2021202775-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-10-07 WO disclosed
US-10174065-B2 Antidiabetic enolic glucoside of phenylpyruvic acid ZADEC APS (DK) 2019-01-08 US disclosed
US-9310681-B2 Negative resist composition and patterning process using same SHIN-ETSU CHEMICAL CO., LTD. (JP) 2016-04-12 US disclosed
US-9310681-B2 Negative resist composition and patterning process using same SHIN-ETSU CHEMICAL CO., LTD. (JP) 2016-04-12 US disclosed
US-20160083411-A1 ANTIDIABETIC ENOLIC GLUCOSIDE OF PHENYLPYRUVIC ACID ZADEC APS (DK) 2016-03-24 US disclosed
WO-2004026293-A2 HEMIASTERLIN DERIVATIVES FOR TREATING RESISTANT TUMORS WYETH HOLDINGS CORPORATION (US) 2004-04-01 WO disclosed
CN-1083422-C Process for production of phenyllatic acid derivative MITSUBISHI ARTIFICIAL SILK CO (JP) 2002-04-24 CN disclosed
EP-0696566-B1 Process for production of phenyllactic acid derivative NITTO CHEMICAL INDUSTRY CO LTD (JP) 1998-06-10 EP disclosed
US-5684186-A HYDROGENATION OF A PHENYLPYRUVIC DERIVATIVE NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1997-11-04 US disclosed
CN-1122325-A Process for production of phenyllatic acid derivative NITTO CHEMICAL INDUSTRY CO LTD (JP) 1996-05-15 CN disclosed
EP-0696566-A1 Process for production of phenyllactic acid derivative NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1996-02-14 EP disclosed
US-4849345-A L-phenylalanine dehydrogenase and use thereof SAGAMI CHEMICAL RESEARCH CENTER (JP) 1989-07-18 US disclosed
EP-0206460-A2 L-phenylalanine dehydrogenase and use thereof SAGAMI CHEMICAL RESEARCH CENTER (JP) 1986-12-30 EP disclosed
US-4220767-A HISTAMINE ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-09-02 US disclosed
US-4185103-A ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-01-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10174065-B2 Antidiabetic enolic glucoside of phenylpyruvic acid PC, SLC5A1, SLC5A2 CTBP2 2912/4885MEN1 3508/4885KMT2A 4011/4885
US-12428403-B2 N-(heterocyclyl and heterocyclylalkyl)-3-benzylpyridin-2-amine derivatives as SSTR4 agonists SSTR4, SSTR3, SSTR1 CTBP2 3844/4885MEN1 397/4885KMT2A 4403/4885
US-20160083411-A1 ANTIDIABETIC ENOLIC GLUCOSIDE OF PHENYLPYRUVIC ACID PC, SLC5A1, SLC5A2 CTBP2 2912/4885MEN1 3508/4885KMT2A 4011/4885
US-20230192659-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS SSTR4, SSTR3, SSTR1 CTBP2 3844/4885MEN1 397/4885KMT2A 4403/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.