SCHEMBL7293162

SCHEMBL7293162

C=C(Cc1cccc(OC)c1)C(=O)O

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTBP2 P56545 1/20 0.64
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
CYP1A2 P05177 1/20 0.54
USP2 O75604 1/20 0.51
POLB P06746 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MMP13 P45452 1/20 0.49
LMNA P02545 1/20 0.49
RAB9A P51151 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27761857 0.86 CTBP2 (0.55) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL6441998 0.84 MEN1 (0.54) CTBP2MEN1KMT2ACYP1A2ALDH1A1
SCHEMBL6499293 0.84 FFAR1 (0.51) CTBP2ALDH1A1SMN1; SMN2LMNA
SCHEMBL6670971 0.83 CTBP2 (0.68) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL29824310 0.83 PTGS1 (0.67) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL229067 0.83 PTGS1 (0.67) CTBP2MEN1KMT2ACYP1A2USP2
SCHEMBL3423556 0.82 CTBP2 (0.44) CTBP2CYP1A2
SCHEMBL29846895 0.82 CTBP2 (0.51) CTBP2MEN1KMT2ACYP1A2POLB
SCHEMBL1621499 0.82 HDAC1 (0.58) CTBP2MEN1KMT2ACYP1A2ALDH1A1
SCHEMBL7341455 0.82 CTBP2 (0.51) CTBP2MEN1KMT2ACYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109369637-A The novel derivative of kojic acid of one kind thiadiazoles containing 1,3,4- and its application 湖南科技大学 2019-02-22 CN disclosed
EP-0636621-B1 Beta-mercapto-propanamide derivatives useful in the treatment of cardiovascular diseases ZAMBON SPA (IT) 1997-03-12 EP disclosed
US-5506259-A β-mercapto-propanamide derivatives useful in the treatment of cardiovascular diseases ZAMBON GROUP S.P.A. (IT) 1996-04-09 US disclosed
US-5389616-A Renin inhibitor, hypotensive agent HOFFMAN-LAROCHE INC. (US) 1995-02-14 US disclosed
EP-0636621-A1 Beta-mercapto-propanamide derivatives useful in the treatment of cardiovascular diseases ZAMBON GROUP S.p.A. (IT) 1995-02-01 EP disclosed
US-5256645-A Renin inhibitors; hypotensive agents HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US disclosed
US-5134123-A Renin enzyme inhibitors for cardiovascular disorders and high blood pressure HOFFMAN-LA ROCHE INC. (US) 1992-07-28 US disclosed
EP-0332008-A2 Peptide-like aminoacid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-09-13 EP disclosed