SCHEMBL6671464

SCHEMBL6671464

Cc1ccc2nc(-c3ccc(Br)cc3)nc(C(N)C3CCCCC3)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.38
RAB9A P51151 5/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
HTT P42858 2/20 0.38
XBP1 P17861 1/20 0.38
ATM Q13315 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TP53 P04637 2/20 0.37
CYP1A1 P04798 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP1B1 Q16678 2/20 0.36
PDE5A O76074 2/20 0.36
ACP1 P24666 2/20 0.36
MC4R P32245 1/20 0.36
MAPT P10636 3/20 0.35
SLC6A3 Q01959 1/20 0.35
MAPK1 P28482 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3977120 0.88 NPC1 (0.49) NPC1RAB9AL3MBTL1HTTATM
SCHEMBL3976890 0.83 SLC2A1 (0.46) NPSR1
SCHEMBL3974312 0.74 POLB (0.53) NPC1RAB9AL3MBTL1HTTNPSR1
SCHEMBL3973240 0.74 HTT (0.43) NPC1RAB9AHTTXBP1ATM
SCHEMBL3978931 0.74 KCNH2 (0.42) NPC1RAB9AHTTXBP1ATM
SCHEMBL27599318 0.74 TP53 (0.39) NPC1RAB9AL3MBTL1HTTXBP1
SCHEMBL3974310 0.73 GBA1 (0.51) PDE5AKMT2A
SCHEMBL3973898 0.70 LMNA (0.45) NPC1RAB9AHTTXBP1ATM
SCHEMBL27581755 0.69 SLC6A3 (0.41) NPC1RAB9AL3MBTL1HTTXBP1
SCHEMBL3979623 0.68 POLB (0.37) TP53CYP1A1CYP1A2CYP1B1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004030672-A1 USE OF 4 AMINO-QUINAZOLINES AS ANTI CANCER AGENTS MERCK PATENT GMBH (DE) 2004-04-15 WO disclosed