SCHEMBL6672730

SCHEMBL6672730

Clc1nc(Cl)nc(NCCc2ccccc2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.60
CA1 P00915 3/20 0.60
CA2 P00918 3/20 0.60
CA9 Q16790 3/20 0.60
CA14 Q9ULX7 3/20 0.60
APP P05067 3/20 0.59
KCNH3 Q9ULD8 1/20 0.51
BCHE P06276 1/20 0.50
ACHE P22303 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50
CA7 P43166 1/20 0.50
CA13 Q8N1Q1 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 2/20 0.49
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20511434 0.89 HPGD (0.62) CA12CA1CA2CA9CA14
SCHEMBL10851721 0.88 HPGD (0.56) CA12CA1CA2CA9CA14
SCHEMBL22151175 0.86 APP (0.64) APPKCNH3BCHEACHEL3MBTL1
SCHEMBL7024590 0.84 APP (0.54) APPKCNH3BCHEACHEL3MBTL1
SCHEMBL1309478 0.84 CA12 (0.59) CA12CA1CA2CA9CA14
SCHEMBL1562297 0.82 APP (0.59) CA12CA1CA2CA9CA14
SCHEMBL6673861 0.82 APP (0.47) CA12CA1CA2CA9CA14
SCHEMBL6674407 0.82 CA9 (0.61) CA12CA1CA2CA9CA14
SCHEMBL1312011 0.82 PKM (0.66) CA12CA1CA2CA9CA14
SCHEMBL8347870 0.80 HDAC1 (0.56) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108191774-B Heterocyclic compound, preparation method and application thereof 中国药科大学 2022-05-24 CN disclosed
WO-2020146779-A1 mTORC1 INHIBITORS FOR ACTIVATING AUTOPHAGY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-07-16 WO disclosed
WO-2018175958-A1 THIOREDOXIN MODULATORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-09-27 WO disclosed
WO-2004035199-A1 AFFINITY ADSORBENTS FOR IMMUNOGLOBULINS CAMBRIDGE UNIVERSITY TECHNICAL SERVICES LIMITED (GB) 2004-04-29 WO disclosed