SCHEMBL6672732

SCHEMBL6672732

NC(=O)c1ccnc(-c2nccs2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.43
HSP90AA1 P07900 1/20 0.42
MYC P01106 1/20 0.41
ECE1 P42892 1/20 0.40
ADORA2A P29274 2/20 0.40
ABL1 P00519 1/20 0.39
BCR P11274 1/20 0.39
TGFBR1 P36897 1/20 0.38
HDAC2 Q92769 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
KDM4B O94953 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6649178 0.81 ECE1 (0.38) CHEK2HSP90AA1MYCECE1ADORA2A
SCHEMBL9081101 0.80 ADORA3 (0.43) KDM4BKDM5CKDM5B
SCHEMBL6646535 0.76 AURKA (0.48) CHEK2ADORA2ACYP3A4HPGD
SCHEMBL13727555 0.75 PARP1 (0.42) CYP3A4
SCHEMBL30416558 0.74 CHEK2 (0.43) CHEK2MYCECE1ADORA2AABL1
SCHEMBL2547481 0.74 HSP90AA1 (0.53) HSP90AA1ADORA2ATGFBR1HDAC2HDAC3
SCHEMBL31122242 0.73 HTR2B (0.51) CHEK2HSP90AA1ECE1ADORA2AHDAC3
SCHEMBL29520114 0.73 CHEK2 (0.44) CHEK2ADORA2AHDAC1HDAC6ADORA1
SCHEMBL18113788 0.73 CHEK2 (0.50) CHEK2HSP90AA1MYCECE1ADORA2A
SCHEMBL2592323 0.71 CHEK2 (0.68) CHEK2MYCABL1BCRTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012151567-A1 PYRIMIDINONE COMPOUNDS AND METHODS FOR PREVENTING AND TREATING INFLUENZA ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2012-11-08 WO disclosed
EP-1441734-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2004-08-04 EP disclosed
WO-2003035076-A1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2003-05-01 WO disclosed