SCHEMBL667329

SCHEMBL667329

COc1ccc(CNC(=O)c2cc(Cl)nnc2Cl)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.58
ALDH1A1 P00352 3/20 0.57
APEX1 P27695 1/20 0.56
RAB9A P51151 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.52
HPGD P15428 1/20 0.52
HCRTR1 O43613 2/20 0.52
HCRTR2 O43614 2/20 0.52
HTR1A P08908 1/20 0.52
OPRM1 P35372 1/20 0.52
DRD3 P35462 1/20 0.52
HTR2B P41595 1/20 0.52
KCNH2 Q12809 1/20 0.52
KMT2A Q03164 2/20 0.51
TSHR P16473 1/20 0.51
MAPK10 P53779 1/20 0.51
MEN1 O00255 1/20 0.51
NOD2 Q9HC29 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30277768 0.83 HCRTR2 (0.68) LMNAALDH1A1APEX1SMN1; SMN2HCRTR1
SCHEMBL664536 0.83 HCRTR2 (0.68) LMNAALDH1A1APEX1SMN1; SMN2HCRTR1
SCHEMBL3623808 0.82 HCRTR1 (0.58) LMNAALDH1A1APEX1SMN1; SMN2HCRTR1
SCHEMBL666493 0.81 HCRTR2 (0.71) LMNAALDH1A1APEX1SMN1; SMN2HCRTR1
SCHEMBL667749 0.80 HCRTR2 (0.73) LMNAAPEX1RAB9ASMN1; SMN2HCRTR2
SCHEMBL2276982 0.77 HCRTR2 (0.72) LMNAAPEX1SMN1; SMN2HCRTR1HCRTR2
SCHEMBL28628718 0.76 KMT2A (0.64) ALDH1A1SMN1; SMN2HPGDKMT2AMEN1
SCHEMBL31683865 0.76 KMT2A (0.64) ALDH1A1SMN1; SMN2HPGDKMT2AMEN1
SCHEMBL6942022 0.76 LMNA (0.61) LMNAALDH1A1APEX1SMN1; SMN2HPGD
SCHEMBL8206949 0.75 LMNA (0.57) LMNAALDH1A1APEX1L3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12414565-B2 Pyridazine (THIO)amides as fungicidal compounds BAYER AKTIENGESELLSCHAFT (DE) 2025-09-16 US disclosed
EP-3887362-B1 PYRIDAZINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AG (DE) 2025-06-18 EP disclosed
US-20230054449-A1 PYRIDAZINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2023-02-23 US disclosed
EP-2349267-B1 PYRIDAZINE CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2014-06-25 EP disclosed
EP-2349267-B1 PYRIDAZINE CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2014-06-25 EP disclosed
US-8703770-B2 Pyridazine carboxamide orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2014-04-22 US disclosed
US-8703770-B2 Pyridazine carboxamide orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2014-04-22 US disclosed
US-8703770-B2 Pyridazine carboxamide orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2014-04-22 US disclosed
US-20120046289-A1 Pyridazine Carboxamide Orexin Receptor Antagonists MERCK SHARP & DOHME CORP. 2012-02-23 US disclosed
US-20120046289-A1 Pyridazine Carboxamide Orexin Receptor Antagonists MERCK SHARP & DOHME CORP. 2012-02-23 US disclosed
US-20120046289-A1 Pyridazine Carboxamide Orexin Receptor Antagonists MERCK SHARP & DOHME CORP. 2012-02-23 US disclosed
EP-2349267-A1 PYRIDAZINE CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2011-08-03 EP disclosed
WO-2010051238-A1 PYRIDAZINE CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-05-06 WO disclosed
WO-2010051238-A1 PYRIDAZINE CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12414565-B2 Pyridazine (THIO)amides as fungicidal compounds PNPO, TPMT, BLVRB LMNA 3826/4885ALDH1A1 2326/4885APEX1 709/4885
US-20120046289-A1 Pyridazine Carboxamide Orexin Receptor Antagonists HCRTR2, HCRTR1, NPY5R LMNA 2800/4885ALDH1A1 3353/4885APEX1 4779/4885
US-20230054449-A1 PYRIDAZINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS PNPO, TPMT, BLVRB LMNA 4608/4885ALDH1A1 2740/4885APEX1 1245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.