SCHEMBL6673318

SCHEMBL6673318

Cc1ccncc1-c1nccs1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 10/20 0.65
CYP2A6 P11509 4/20 0.49
CYP1A2 P05177 8/20 0.48
PDPK1 O15530 1/20 0.41
CYP2E1 P05181 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2B6 P20813 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP2C8 P10632 2/20 0.41
ABL1 P00519 1/20 0.39
ADRB2 P07550 1/20 0.38
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
SRC P12931 1/20 0.37
ZAP70 P43403 1/20 0.37
SYK P43405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6629919 0.82 CYP17A1 (0.55) CYP17A1CYP2A6CYP1A2CYP2E1CYP3A4
SCHEMBL14830742 0.80 CYP17A1 (1.00) CYP17A1CYP2A6CYP1A2
SCHEMBL6630051 0.79 CYP17A1 (0.52) CYP17A1CYP2A6CYP1A2CYP2E1CYP3A4
SCHEMBL1047236 0.77 PDPK1 (0.53) CYP17A1CYP2A6CYP1A2PDPK1CYP3A4
SCHEMBL6630189 0.76 CYP17A1 (0.49) CYP17A1CYP2A6CYP1A2
SCHEMBL2588012 0.75 CYP17A1 (0.69) CYP17A1CYP1A2
SCHEMBL3421743 0.75 TDO2 (0.49) CYP17A1CYP2A6CYP1A2CYP2E1CYP3A4
SCHEMBL29988790 0.75 TDO2 (0.49) CYP17A1CYP2A6CYP1A2CYP2E1CYP3A4
SCHEMBL1290082 0.74 SRC (0.50) CYP17A1CYP2A6CYP1A2PDPK1CYP3A4
SCHEMBL10053508 0.74 CYP1A2 (0.44) CYP17A1CYP2A6CYP1A2CYP2E1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019149260-A1 PYRIDAZINOL COMPOUND, DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR, HERBICIDAL COMPOSITION AND USE THEREOF 青岛清原化合物有限公司 2019-08-08 WO disclosed
EP-1432706-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
WO-2003027085-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed