SCHEMBL6630189

SCHEMBL6630189

COc1cccc(-c2cnccc2C)c1-c1nccs1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 16/20 0.49
CYP1A2 P05177 10/20 0.47
BDKRB2 P30411 1/20 0.39
CYP2A6 P11509 1/20 0.38
SMPD3 Q9NY59 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6673318 0.76 CYP17A1 (0.65) CYP17A1CYP1A2CYP2A6
SCHEMBL1988909 0.74 FYN (0.43) SMPD3
SCHEMBL5085483 0.73 SMPD3 (0.45) CYP1A2SMPD3
SCHEMBL26259608 0.72 SMPD3 (0.42) CYP1A2BDKRB2SMPD3
SCHEMBL5396495 0.72 ADRA1D (0.52) CYP1A2SMPD3
SCHEMBL29715238 0.72 ADRA1D (0.52) CYP1A2SMPD3
SCHEMBL2152304 0.71 GAA (0.54) CYP1A2SMPD3
SCHEMBL14830909 0.70 CYP17A1 (0.65) CYP17A1CYP1A2
SCHEMBL26259637 0.69 SMPD3 (0.50) CYP2A6SMPD3
SCHEMBL3201031 0.68 PARP1 (0.46) SMPD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432706-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
WO-2003027085-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed