SCHEMBL6674009

SCHEMBL6674009

O=C1c2c(O)ccc(O)c2C(=O)c2c(Cl)ccc(F)c21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 3/20 0.44
CSNK2B P67870 3/20 0.44
CSNK2A1 P68400 3/20 0.44
CSNK2A3 Q8NEV1 3/20 0.44
CYP3A4 P08684 4/20 0.43
HPGD P15428 4/20 0.43
TSHR P16473 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TP53 P04637 2/20 0.43
HIF1A Q16665 1/20 0.43
MAPT P10636 5/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
MAPK1 P28482 4/20 0.41
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 4/20 0.41
TDP1 Q9NUW8 4/20 0.41
MAOA P21397 3/20 0.41
KDM4E B2RXH2 2/20 0.41
USP2 O75604 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3896954 0.88 CSNK2A2 (0.54) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL7738621 0.88 CSNK2A2 (0.54) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL30887225 0.88 CSNK2A2 (0.54) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL10356073 0.88 CSNK2A2 (0.54) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL497611 0.88 CSNK2A2 (0.54) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL1323063 0.88 CSNK2A2 (0.54) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL7742020 0.88 CSNK2A2 (0.54) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL9059735 0.85 CSNK2A2 (0.44) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL11852041 0.80 CSNK2A2 (0.47) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4
SCHEMBL11156531 0.78 GPR55 (0.45) CSNK2A2CSNK2BCSNK2A1CSNK2A3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1097125-B1 PROCESS FOR THE PREPARATION OF 1,4-BIS[[2-(DIMETHYLAMINO)ETHYL AMINO]-5,8-DIHYDROXYANTHRACENE-9,10-DIONE BTG INTERNAT LTD COMPANY NO 26 (GB) 2004-09-29 EP disclosed
US-6320063-B1 HEATING DICHLOROPHTHALIC ANHYDRIDE OVER LAYER OF POWDERED ANHYDROUS SODIUM AND/OR POTASSIUM FLUORIDE UNDER NITROGEN ATMOSPHERE TO PRODUCE DIFLUOROPHTHALIC ANHYDRIDE INTERMEDIATE BTG INTERNATIONAL LIMITED (GB) 2001-11-20 US disclosed
EP-1097125-A1 PROCESS FOR THE PREPARATION OF 1,4-BIS[[2-(DIMETHYLAMINO)ETHYL AMINO]-5,8-DIHYDROXYANTHRACENE-9,10-DIONE BTG INTERNATIONAL LIMITED (Company No. 2664412) (GB) 2001-05-09 EP disclosed
WO-2000005194-A1 PROCESS FOR THE PREPARATION OF 1,4-BIS[[2- (DIMETHYLAMINO) ETHYL] AMINO] -5,8- DIHYDROXYANTHRACENE- 9,10-DIONE BTG INTERNATIONAL LIMITED (GB) 2000-02-03 WO disclosed