Dioxybenzone

Dioxybenzone

SCHEMBL6674075

COc1ccc(C(=O)c2ccccc2O)c(O)c1.COc1ccc(C(=O)c2ccccc2O)c(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 1.00
CYP2C19 P33261 4/20 1.00
HPGD P15428 3/20 1.00
CYP3A4 P08684 3/20 1.00
CYP1A2 P05177 2/20 1.00
PGR P06401 2/20 1.00
SLC6A2 P23975 2/20 1.00
ADORA3 P0DMS8 1/20 1.00
AR P10275 1/20 1.00
CHRM1 P11229 1/20 1.00
ALOX15 P16050 1/20 1.00
TBXA2R P21731 1/20 1.00
ADRA1A P35348 1/20 1.00
HIF1A Q16665 1/20 1.00
NPC1 O15118 7/20 0.83
RAB9A P51151 6/20 0.83
MAPK1 P28482 3/20 0.73
ALDH1A1 P00352 2/20 0.73
CYP2D6 P10635 2/20 0.73
PDE4A P27815 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dioxybenzone SCHEMBL29364693 1.00 LMNA (1.00) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL7936480 1.00 LMNA (1.00) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL29354139 1.00 LMNA (1.00) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL15894 1.00 LMNA (1.00) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL29365575 1.00 LMNA (1.00) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL20641426 0.97 LMNA (0.94) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL5011376 0.95 HPGD (0.91) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL5161579 0.92 HPGD (0.88) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL4923214 0.92 HPGD (0.88) LMNACYP2C19HPGDCYP3A4CYP1A2
Dioxybenzone SCHEMBL28167789 0.92 HPGD (0.85) LMNACYP2C19HPGDCYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013102248-A2 \"AQUEOUS COSMETIC SUNSCREEN COMPOSITION AND USE THEREOF, COSMETIC METHOD FOR APPLICATION OF SAID COMPOSITION, COSMETIC METHOD TO PREVENT AND CONTROL SKIN OILINESS, COSMETIC METHOD TO PROTECT THE SKIN FROM THE DAMAGES CAUSED BY ULTRAVIOLET RADIATION, AND COSMETIC PRODUCT.\ . JOHNSON & JOHNSON DO BRASIL INDUSTRIA E COMERCIO DE PRODUTOS PARA SAUDE LTDA. (BR) 2013-07-11 WO claimed
EP-3651732-A1 LIGHT AESTHETIC SUNSCREEN COMPOSITIONS Johnson & Johnson Consumer Inc. (US) 2020-05-20 EP disclosed
EP-3481365-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2019-05-15 EP disclosed
EP-3471694-A1 SUNSCREEN COMPOSITIONS CONTAINING A COMBINATION OF A LINEAR ULTRAVIOLET RADIATION-ABSORBING POLYETHER AND OTHER ULTRAVIOLET-SCREENING COMPOUNDS Johnson & Johnson Consumer Inc. (US) 2019-04-24 EP disclosed
WO-2019014568-A1 LIGHT AESTHETIC SUNSCREEN COMPOSITIONS JOHNSON & JOHNSON CONSUMER INC. (US) 2019-01-17 WO disclosed
WO-2018007577-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2018-01-11 WO disclosed
WO-2017218390-A1 SUNSCREEN COMPOSITIONS CONTAINING A COMBINATION OF A LINEAR ULTRAVIOLET RADIATION-ABSORBING POLYETHER AND OTHER ULTRAVIOLET-SCREENING COMPOUNDS JOHNSON & JOHNSON CONSUMER INC. (US) 2017-12-21 WO disclosed
EP-3229766-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2017-10-18 EP disclosed
EP-3128995-A1 SOLUBLIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2017-02-15 EP disclosed
EP-3041904-A1 STYRYL SULFIDE DYES BASF SE (DE) 2016-07-13 EP disclosed
WO-2003051375-A1 STABILIZED BRIVUDINE TOPICAL FORMULATIONS MENARINI RICERCHE S.P.A. (IT) 2003-06-26 WO disclosed
EP-1318720-A2 ANTIMICROBIAL TERNARY SURFACTANT BLEND COMPRISING CATIONIC, ANIONIC, AND BRIDGING SURFACTANTS, AND METHODS OF PREPARING SAME STEPAN COMPANY (US) 2003-06-18 EP disclosed
WO-2002022083-A2 EMULSION COMPRISING A BLEND OF CATIONIC, ANIONIC AND BRIDGING SURFACTANTS, OIL AND WATER STEPAN COMPANY (US) 2002-03-21 WO disclosed
WO-2002021916-A2 ANTIMICROBIAL TERNARY SURFACTANT BLEND COMPRISING CATIONIC, ANIONIC, AND BRIDGING SURFACTANTS, AND METHODS OF PREPARING SAME STEPAN COMPANY (US) 2002-03-21 WO disclosed
US-6143906-A REACTING ASCORBIC ACID OR ASCORBIC ACID DERIVATIVES WITH SORBIC ACID OR SORBIC ACID DERIVATIVE TO FORM ASCORBYL SORBATES WHICH IS USED AS COSMETIC OR DURG BASF AKTIENGESELLSCHAFT (DE) 2000-11-07 US disclosed
US-6069258-A SUNSCREEN AGENTS; PROTECTIVE COATINGS FOR SKIN BASF AKTIENGESELLSCHAFT (DE) 2000-05-30 US disclosed
US-6007828-A SUNSCREEN AGENT MIXTURE CONTAINING 1,1-DINITRILO-2,2-DIPHENYL ETHYLENE DERIVATIVE IN A COSMETIC CARRIER BASF AKTIENGESELLSCHAFT (DE) 1999-12-28 US disclosed
US-5968484-A APPLYING 2-ORGANOCARBONYLACRYLONITRILE DERIVATIVE AS SUNSCREEN AGENT BASF AKTIENGESELLSCHAFT (DE) 1999-10-19 US disclosed
EP-0814760-A1 SUBSTITUTED o-AMINOCARBONYLBENZOIC ACID SALTS AND THEIR USE AS SUNSCREENS STEPAN COMPANY (US) 1998-01-07 EP disclosed
WO-1997025971-A1 SUBSTITUTED o-AMINOCARBONYLBENZOIC ACID SALTS AND THEIR USE AS SUNSCREENS STEPAN COMPANY (US) 1997-07-24 WO disclosed