SCHEMBL6674186

SCHEMBL6674186

NC(=O)C1CN(c2ccc(N3Cc4cccnc4C3)c(F)c2)C(=O)O1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 8/20 0.49
MAOB P27338 10/20 0.42
CALML3 P27482 2/20 0.41
LMNA P02545 1/20 0.41
PTGS1 P23219 1/20 0.41
SDHA P31040 1/20 0.41
TIPARP Q7Z3E1 1/20 0.39
F10 P00742 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3036235 1.00 MAOA (0.49) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL5765558 0.93 MAOB (0.42) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL3038203 0.89 MAOB (0.43) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL3041156 0.89 MAOB (0.43) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL6636437 0.86 CALML3 (0.56) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL6638114 0.82 MAOA (0.65) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL6672496 0.81 TIPARP (0.38) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL6208782 0.78 MAOA (0.58) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL13515442 0.78 MAOA (0.58) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL3041159 0.77 TIPARP (0.39) MAOAMAOBCALML3LMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645781-B2 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PFIZER INC (US) 2010-01-12 US disclosed
EP-1478629-A1 N-ARYL-2-OXAZOLIDINONE-5-CARBOXAMIDES AND THEIR DERIVATIVES AND THEIR USE AS ANTIBACTERIALS PHARMACIA & UPJOHN COMPANY (US) 2004-11-24 EP disclosed
WO-2003072553-A1 N-ARYL-2-OXAZOLIDINONE-5-CARBOXAMIDES AND THEIR DERIVATES AND THEIR USE AS ANTIBACTERIALS PHARMACIA & UPJOHN COMPANY (US) 2003-09-04 WO disclosed