SCHEMBL6674535

SCHEMBL6674535

N#Cc1ccccc1-c1c(-c2ccccc2)c(-c2ccc(O)cn2)c[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.40
MCL1 Q07820 3/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
DYRK1A Q13627 1/20 0.37
FASN P49327 2/20 0.36
GALR3 O60755 1/20 0.35
GAA P10253 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
PIM1 P11309 2/20 0.34
BIRC5 O15392 1/20 0.34
CHEK1 O14757 1/20 0.34
WEE1 P30291 1/20 0.34
LRRK2 Q5S007 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3672706 0.87 KDM4E (0.40) MCL1KDM4EALDH1A1HPGDGABRG2
SCHEMBL2918049 0.84 GRIA1 (0.47) MCL1KDM4EALDH1A1HPGDGABRG2
Water SCHEMBL4777584 0.84 GRIA1 (0.47) MCL1KDM4EALDH1A1HPGDGABRG2
SCHEMBL6680176 0.80 LRRK2 (0.44) ESR2MCL1KDM4EALDH1A1HPGD
SCHEMBL6686812 0.80 GRIA1 (0.47) MCL1KDM4EALDH1A1HPGDGABRG2
SCHEMBL6695728 0.79 MCL1 (0.45) MCL1KDM4EALDH1A1HPGDGABRG2
SCHEMBL6693263 0.79 MCL1 (0.40) MCL1KDM4EALDH1A1HPGDGABRG2
SCHEMBL3667255 0.78 PIM1 (0.41) ESR2MCL1KDM4EALDH1A1HPGD
SCHEMBL3666760 0.78 MCL1 (0.41) MCL1KDM4EALDH1A1HPGDGABRG2
SCHEMBL3677714 0.77 TGFBR1 (0.42) MCL1KDM4EALDH1A1HPGDGABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed