SCHEMBL6674686

SCHEMBL6674686

FC(F)(F)c1ccc(N2CCNCC2)cc1.O=S(=O)(Cl)N1CCN(c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.53
ADRB1 P08588 3/20 0.50
HTR6 P50406 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HTR3E A5X5Y0 2/20 0.49
HTR3B O95264 2/20 0.49
HTR3A P46098 2/20 0.49
HTR3D Q70Z44 2/20 0.49
HTR3C Q8WXA8 2/20 0.49
SIGMAR1 Q99720 2/20 0.49
HTR1D P28221 1/20 0.49
HTR2C P28335 1/20 0.49
MAPT P10636 1/20 0.48
THRB P10828 1/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.47
CA12 O43570 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4700945 0.91 CA2 (0.54) ALDH1A1THRBGAACA12CA2
SCHEMBL7178620 0.84 ADRB1 (0.67) MAOBADRB1HTR6ALDH1A1HTR3E
SCHEMBL233850 0.84 ADRB1 (0.67) MAOBADRB1HTR6ALDH1A1HTR3E
Hydrochloric Acid SCHEMBL29882384 0.83 MAPT (0.65) MAOBADRB1HTR6ALDH1A1HTR3E
Hydrochloric Acid SCHEMBL2961970 0.83 MAPT (0.65) MAOBADRB1HTR6ALDH1A1HTR3E
SCHEMBL7474849 0.80 ADRB1 (0.61) MAOBADRB1HTR6ALDH1A1HTR3E
SCHEMBL5239716 0.79 ADRB1 (0.59) MAOBADRB1HTR6ALDH1A1HTR3E
SCHEMBL6242244 0.79 CA2 (0.54) THRBGAACA12CA2CA9
SCHEMBL2156809 0.77 KDM4E (0.55) ALDH1A1MAPTTHRBKDM4EGAA
SCHEMBL4698660 0.77 CA2 (0.56) THRBGAACA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444202-A1 NOVEL METALLOPROTEINASE INHIBITORS AstraZeneca AB (SE) 2004-08-11 EP disclosed
WO-2003040098-A1 NOVEL METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2003-05-15 WO disclosed