SCHEMBL6675145

SCHEMBL6675145

CC(c1cccc([N+](=O)[O-])c1)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
AURKA O14965 1/20 0.47
RPS6KB1 P23443 1/20 0.47
MEN1 O00255 1/20 0.47
HPGD P15428 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPT P10636 3/20 0.46
RAB9A P51151 2/20 0.46
ALOX5 P09917 1/20 0.46
NPC1 O15118 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPY5R Q15761 1/20 0.43
CYP26A1 O43174 1/20 0.42
ACP3 P15309 1/20 0.42
ALDH1A1 P00352 3/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 2/20 0.42
NR3C2 P08235 1/20 0.42
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28468881 0.88 KMT2A (0.45) KMT2AAURKARPS6KB1MEN1HPGD
SCHEMBL3903609 0.83 AURKA (0.45) KMT2AAURKARPS6KB1MEN1HPGD
SCHEMBL665633 0.81 AURKA (0.57) KMT2AAURKARPS6KB1MEN1HPGD
SCHEMBL11092415 0.80 MAPT (0.48) KMT2AMEN1HPGDL3MBTL1MAPT
SCHEMBL31226523 0.79 ACHE (0.43) ALOX5
SCHEMBL6675085 0.79 ACHE (0.43) ALOX5
SCHEMBL29868333 0.77 ALDH1A1 (0.49) KMT2AMEN1MAPTRAB9AALOX5
SCHEMBL3913255 0.77 ALDH1A1 (0.49) KMT2AMEN1MAPTRAB9AALOX5
SCHEMBL2379533 0.77 ANPEP (0.42) HPGDMAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL2378736 0.77 ANPEP (0.42) HPGDMAPTSMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed