SCHEMBL6676446

SCHEMBL6676446

COC(=O)c1[nH]c(=O)ccc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.48
EGFR P00533 1/20 0.47
ALDH1A1 P00352 5/20 0.45
LMNA P02545 3/20 0.45
GAA P10253 2/20 0.45
FGFR1 P11362 1/20 0.45
SRC P12931 1/20 0.45
FGFR2 P21802 1/20 0.45
FGFR4 P22455 1/20 0.45
FGFR3 P22607 1/20 0.45
KDM4E B2RXH2 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
PADI4 Q9UM07 1/20 0.45
GABRA1 P14867 2/20 0.43
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
GABRA3 P34903 2/20 0.43
ERCC1 P07992 1/20 0.43
FEN1 P39748 1/20 0.43
ERCC4 Q92889 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16007019 0.77 HTT (0.54) HTTEGFRALDH1A1LMNAGAA
SCHEMBL3640867 0.74 NR4A2 (0.47) ALDH1A1LMNAGAAFGFR1SRC
SCHEMBL16631726 0.74 CHEK1 (0.45) HTTALDH1A1GAAKDM4ENPSR1
SCHEMBL10465981 0.74 KDM4E (0.53) HTTALDH1A1LMNAGAAKDM4E
SCHEMBL13228930 0.73 HTT (0.62) HTTEGFRALDH1A1LMNAFGFR1
SCHEMBL19669163 0.72 ALDH1A1 (0.55) HTTALDH1A1LMNAGAAFGFR1
SCHEMBL2651508 0.72 TSHR (0.49) HTTALDH1A1LMNAGAAKDM4E
SCHEMBL689403 0.71 PTGER2 (0.60) ALDH1A1LMNAKDM4ENPSR1GABRA1
SCHEMBL21056612 0.70 NR4A2 (0.56) HTTEGFRALDH1A1GAAFGFR1
SCHEMBL11010732 0.70 PDE4A (0.53) HTTALDH1A1GAAKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed