SCHEMBL6676644

SCHEMBL6676644

Cn1c(=O)[nH]c(=O)c2c1nc(N1CCCC(N)C1)n2Cc1cccc(F)c1.NC1CCCN(c2nc3c(c(=O)[nH]c(=O)n3Cc3ccccc3)n2Cc2ccccc2OC(F)F)C1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
TSHR P16473 5/20 0.53
HSD17B10 Q99714 2/20 0.53
THRB P10828 1/20 0.53
NPSR1 Q6W5P4 3/20 0.51
HTT P42858 3/20 0.51
DPP4 P27487 11/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
ALOX15 P16050 1/20 0.49
GAA P10253 1/20 0.48
USP2 O75604 1/20 0.47
MAPT P10636 2/20 0.47
MAPK1 P28482 2/20 0.47
POLB P06746 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4667805 0.90 DPP4 (0.52) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL4668769 0.87 ALDH1A1 (0.59) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL4668509 0.86 DPP4 (0.57) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL4668663 0.82 TSHR (0.73) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL4668748 0.81 DPP4 (0.56) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL4669779 0.80 DPP4 (0.58) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL6674513 0.80 DPP4 (0.66) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL4668968 0.80 ALDH1A1 (0.56) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL4666981 0.80 TSHR (0.72) ALDH1A1TSHRHSD17B10THRBNPSR1
SCHEMBL4668818 0.79 DPP4 (0.66) ALDH1A1TSHRHSD17B10THRBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004033455-A2 HEMISUCCINATE SALTS OF HETEROCYCLIC DPP-IV INHIBITORS NOVO NORDISK A/S (DK) 2004-04-22 WO disclosed