SCHEMBL6677

SCHEMBL6677

CCN(CC)CCOC(=O)c1ccc(NCl)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.67
TSHR P16473 3/20 0.67
MAOA P21397 3/20 0.67
CYP2D6 P10635 3/20 0.67
HTR3A P46098 1/20 0.67
BLM P54132 2/20 0.65
NPSR1 Q6W5P4 1/20 0.65
LMNA P02545 5/20 0.63
SCN1A P35498 4/20 0.63
SCN2A Q99250 4/20 0.63
SCN3A Q9NY46 4/20 0.63
ATM Q13315 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
ALDH1A1 P00352 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
MAPT P10636 2/20 0.53
CYP1A2 P05177 3/20 0.51
KCNH2 Q12809 3/20 0.51
SIGMAR1 Q99720 2/20 0.51
SLC6A3 Q01959 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL8171709 0.99 HRH3 (0.65) HRH3TSHRMAOACYP2D6HTR3A
Hydrochloric Acid SCHEMBL24097 0.99 BLM (0.68) HRH3TSHRMAOACYP2D6HTR3A
Choline SCHEMBL3808986 0.90 HRH3 (0.55) HRH3TSHRMAOACYP2D6HTR3A
SCHEMBL94128 0.87 HRH3 (0.68) HRH3TSHRMAOACYP2D6HTR3A
SCHEMBL4295410 0.87 HRH3 (0.68) HRH3TSHRMAOACYP2D6HTR3A
SCHEMBL3840896 0.86 SMN1; SMN2 (0.53) HRH3TSHRMAOACYP2D6HTR3A
SCHEMBL9576578 0.85 HRH3 (0.71) HRH3TSHRMAOACYP2D6HTR3A
SCHEMBL6616028 0.84 TSHR (0.52) HRH3TSHRMAOACYP2D6HTR3A
SCHEMBL174306 0.84 MAOA (0.49) HRH3TSHRMAOACYP2D6HTR3A
Iodide SCHEMBL1022754 0.84 HRH3 (0.65) HRH3TSHRMAOACYP2D6HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 53508 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144801-A1 COMPOSITIONS AND METHODS FOR PREVENTING OR TREATING MUSCLE CONDITIONS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-05-28 US claimed
EP-4746863-A1 ENDOXIFEN COMPOSITIONS AND METHODS OF USE THEREOF AND SYNTHESIS THEREOF Atossa Therapeutics, Inc. (US) 2026-05-27 EP claimed
US-20260137637-A1 ANESTHETIC AGENT MICRO AND NANO PARTICLES, AND METHODS OF MAKING AND USING THE SAME HAAS ERIC (US) 2026-05-21 US claimed
WO-2026099533-A1 TREATMENT OF ACUTE RESPIRATORY DISTRESS SYNDROME (ARDS) WITH GPBP1 INHIBITORS UNIVERSITAT DE VALÈNCIA (ES) 2026-05-15 WO claimed
WO-2026101937-A1 COMPOSITIONS COMPRISING (Z)-ENDOXIFEN AND A CDK4/6 INHIBITOR AND METHODS OF USE THEREOF ATOSSA THERAPEUTICS, INC. (US) 2026-05-15 WO claimed
US-12622873-B2 Composition of matter comprising liposomes embedded in a polymeric matrix and methods of using same YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2026-05-12 US claimed
EP-4735042-A1 MERCERIZED DECELLULARIZED PARTICLES FOR SLOW RELEASE APPLICATIONS AND METHODS THEREOF Spiderwort Biotechnologies Inc. (CA) 2026-05-06 EP claimed
US-20260115156-A1 INJECTABLE COMPOSITION INCLUDING HYDROGEL CONTAINING ANESTHETIC AGENT UNIV KOREA RES & BUS FOUND (KR) 2026-04-30 US claimed
EP-3723819-B1 WOUND DRESSING ANIMAL ETHICS PTY LTD (AU) 2026-04-22 EP claimed
US-20260097044-A1 ION PAIR LIQUID CRYSTAL FORMULATIONS FOR LONG-ACTING INJECTABLES OF POORLY SOLUBLE DRUGS FORDOZ PHARMA CORP. (US) 2026-04-09 US claimed
EP-0336901-A2 Anesthetic skin moisturizing composition and method of preparing same WARNER-LAMBERT COMPANY (US) 1989-10-11 EP claimed
EP-0331392-A2 Anesthesia and antisepsis of the skin ALZA CORPORATION (US) 1989-09-06 EP claimed
US-4853212-A REMEDIES FOR TREATING SORE THROAT; HEXYLRESOURCINOL WARNER-LAMBERT COMPANY (US) 1989-08-01 US claimed
US-4822597-A FOR THROAT, MOUTH; SWEETENER-ANESTHETIC PREMIX WARNER-LAMBERT COMPANY (US) 1989-04-18 US claimed
EP-0299923-A2 Anesthetic-containing chewing gum compositions WARNER-LAMBERT COMPANY (US) 1989-01-18 EP claimed
EP-0299924-A2 Reduced base content chewing gum compositions having anesthetic properties WARNER-LAMBERT COMPANY (US) 1989-01-18 EP claimed
US-4557934-A ALONG WITH A DIOL PYRROLIDONE OR AN AZACYCLOPENTAN-2-ONE THE PROCTER & GAMBLE COMPANY (US) 1985-12-10 US claimed
US-4495174-A TIME-RELEASE AGENTS RESEARCH CORPORATION (US) 1985-01-22 US claimed
US-4029794-A SAXITOXIN ASTRA PHARMACEUTICAL PRODUCTS, INC. (US) 1977-06-14 US claimed
US-4022899-A TETRODOXIN, DESOXYTETRODOXIN, AMINOALKYL BENZOATE ASTRA PHARMACEUTICAL PRODUCTS, INC. (US) 1977-05-10 US claimed