SCHEMBL6677673

SCHEMBL6677673

COc1cc(C)cc(C(=O)CC(c2ccccc2)S(=O)(=O)O)c1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.44
PDE4B Q07343 2/20 0.44
PDE4C Q08493 2/20 0.44
PDE4D Q08499 2/20 0.44
ALDH1A1 P00352 5/20 0.42
MAPT P10636 5/20 0.42
NPC1 O15118 3/20 0.42
LMNA P02545 3/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TDP1 Q9NUW8 1/20 0.40
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
SRC P12931 1/20 0.38
CTSA P10619 4/20 0.38
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6677057 0.99 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL6677052 0.89 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL6679757 0.76 HTT (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL6675661 0.75 HTT (0.52) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL6679977 0.73 TSHR (0.48) PDE4DALDH1A1MAPTSMN1; SMN2IDO1
SCHEMBL6674306 0.73 SRC (0.46) ALDH1A1MAPTNPC1LMNARAB9A
SCHEMBL6674938 0.72 RAB9A (0.56) ALDH1A1MAPTNPC1LMNARAB9A
SCHEMBL6677164 0.72 SRC (0.45) ALDH1A1MAPTNPC1LMNARAB9A
SCHEMBL6674039 0.71 ALDH1A1 (0.68) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL6674609 0.71 RAB9A (0.55) ALDH1A1MAPTNPC1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204636-B1 3-OXOPROPANE-1-SULPHONIC ACIDS AND SULPHONATES DSM IP ASSETS BV (NL) 2004-10-27 EP disclosed
US-6639103-B1 Enantiomerically enriched forms; resolving amino functiona-lized enantiomers DSM N.V. (NL) 2003-10-28 US disclosed
EP-1204636-A1 3-OXOPROPANE-1-SULPHONIC ACIDS AND SULPHONATES DSM N.V. (NL) 2002-05-15 EP disclosed
WO-2001014327-A1 3-OXOPROPANE-1-SULPHONIC ACIDS AND SULPHONATES DSM N.V. (NL) 2001-03-01 WO disclosed