SCHEMBL6677901

SCHEMBL6677901

O=C(O)C1(C(=O)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.55
SRD5A2 P31213 1/20 0.49
CYP2D6 P10635 3/20 0.48
SLC6A2 P23975 3/20 0.48
SLC6A4 P31645 3/20 0.48
SLC6A3 Q01959 3/20 0.48
KMO O15229 4/20 0.46
PKM P14618 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
MAPT P10636 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
KCNH2 Q12809 1/20 0.46
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15320065 0.84 KMO (0.47) TSHRSRD5A2CYP2D6SLC6A2SLC6A4
SCHEMBL28626237 0.79 TSHR (0.50) TSHRSRD5A2KDM4EMAPTHPGD
SCHEMBL21448794 0.76 TSHR (0.52) TSHRSRD5A2CYP2D6SLC6A2SLC6A4
SCHEMBL21448791 0.76 TSHR (0.52) TSHRSRD5A2CYP2D6SLC6A2SLC6A4
SCHEMBL15319178 0.76 TSHR (0.52) TSHRSRD5A2CYP2D6SLC6A2SLC6A4
SCHEMBL8352471 0.72 TSHR (1.00) TSHRSRD5A2KMOPKMKDM4E
SCHEMBL371998 0.72 TSHR (1.00) TSHRSRD5A2KMOPKMKDM4E
SCHEMBL29353637 0.72 TSHR (1.00) TSHRSRD5A2KMOPKMKDM4E
SCHEMBL4385239 0.72 CES2 (0.46) TSHRKDM4EMEN1NPC1MAPT
SCHEMBL14563971 0.70 MAPT (0.60) TSHRSRD5A2CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1475385-A1 Glycoside derivatives of 2-(3,4-dichlorobenzoyl)-cycopropane-1-carboxylic acid Newron Pharmaceuticals S.p.A. (IT) 2004-11-10 EP disclosed