SCHEMBL6679707

SCHEMBL6679707

COc1ccc(NC(N)=S)c(CCNC(=O)OC(C)(C)C)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.43
MTNR1A P48039 4/20 0.43
MTNR1B P49286 2/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
MAPT P10636 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
DYRK1A Q13627 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6675209 0.83 FAAH (0.40) NQO2MTNR1AMTNR1BCA12CA1
SCHEMBL6675910 0.81 MTNR1A (0.48) NQO2MTNR1AMTNR1BCA12CA1
SCHEMBL6675303 0.80 NQO2 (0.40) NQO2MTNR1AMTNR1BMAPTKDM4E
SCHEMBL6675049 0.80 KMT2A (0.55) CA12CA1CA2CA9MAPT
SCHEMBL29814877 0.80 MTNR1A (0.59) NQO2MTNR1AMTNR1BMAPTRAB9A
SCHEMBL6675304 0.79 MTNR1A (0.41) NQO2MTNR1AMTNR1BMAPTKDM4E
SCHEMBL7239004 0.79 NQO2 (0.41) NQO2MTNR1AMTNR1BCA12CA1
SCHEMBL3152901 0.79 MTNR1A (0.48) NQO2MTNR1AMTNR1BCA12CA1
SCHEMBL5981610 0.79 MTNR1A (0.48) NQO2MTNR1AMTNR1B
SCHEMBL6676121 0.78 CA1 (0.46) NQO2CA1CA2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed