SCHEMBL6679740

SCHEMBL6679740

CC(C)(C)OC(=O)NCc1cccc(NC(N)=N[N+](=O)[O-])c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.46
RPS6KB1 P23443 1/20 0.46
BRD4 O60885 3/20 0.45
CCKBR P32239 1/20 0.42
NAMPT P43490 2/20 0.42
GLS O94925 4/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
SIGMAR1 Q99720 3/20 0.40
GRIN2D O15399 2/20 0.40
GRIN3B O60391 2/20 0.40
GRIN1 Q05586 2/20 0.40
GRIN2A Q12879 2/20 0.40
GRIN2B Q13224 2/20 0.40
GRIN2C Q14957 2/20 0.40
GRIN3A Q8TCU5 2/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6680723 0.90 CYP3A4 (0.45) AURKARPS6KB1NAMPTCA1CA2
SCHEMBL6676314 0.87 NAMPT (0.51) AURKARPS6KB1NAMPTCA1CA2
SCHEMBL6677687 0.84 SIGMAR1 (0.46) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6681977 0.82 AKT1 (0.43) AURKARPS6KB1SIGMAR1GRIN2DGRIN3B
SCHEMBL13162494 0.82 AURKA (0.47) AURKARPS6KB1BRD4CCKBRNAMPT
SCHEMBL6676274 0.82 CA2 (0.41) AURKARPS6KB1CA1CA2SIGMAR1
SCHEMBL6681429 0.81 C5AR1 (0.47) MEN1KMT2A
SCHEMBL7238730 0.81 AURKA (0.46) AURKARPS6KB1BRD4CCKBRNAMPT
SCHEMBL5560988 0.81 AURKA (0.52) AURKARPS6KB1BRD4CCKBRNAMPT
SCHEMBL10209845 0.81 AURKA (0.52) AURKARPS6KB1BRD4CCKBRNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed